A kind of preparation method of acryloyl morpholine
A technology for acryloyl morpholine and morpholine, which is applied in the field of preparing acryloyl morpholine by a single-container method, can solve the problems of serious skin contact or inhalation hazards, difficult separation, hidden safety hazards, etc., and achieves low cost, simple operation, and side reactions. less effect
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Embodiment 1
[0034] Example 1: Preparation of acryloylmorpholine
[0035] In a four-necked flask equipped with a spherical condenser and a stirrer, add 1g p-hydroxyanisole, 21.6g (0.3mol) acrylic acid and 17.7g (0.13mol) phosphorus trichloride, and add 50ml dichloromethane as a solvent , Lower the temperature to 0°C, add 57.4g (0.66mol) of morpholine (previously dissolved in 30ml of dichloromethane) into the reaction solution, slowly add dropwise, control the reaction temperature at 0~5°C, and finish the dropwise addition in 3.5 hours. Incubate the reaction for 1 hour, filter, and spin-dry the solvent to obtain 38 g of crude product, with a GC analysis content of 91%, and vacuum distillation to obtain 34 g with a yield of 81% and a GC content of 99%.
Embodiment 2
[0036] Example 2: Preparation of acryloylmorpholine
[0037] In a four-necked flask equipped with a spherical condenser and stirrer, add 1g phenothiazine, 21.6g (0.3mol) acrylic acid and 17.7g (0.13mol) phosphorus trichloride, and add 50ml of dichloromethane as a solvent to cool down To 0°C, add 57.4g (0.66mol) morpholine (dissolved in 30ml of dichloromethane in advance) to the reaction solution dropwise, slowly add dropwise, control the reaction temperature at 0~5°C, the dropwise addition is over in 3.5 hours, and the reaction is kept warm After 1h, filter and spin-dry the solvent to obtain 37.8g of crude product, GC analysis content is 90%, vacuum distillation obtains 33.2g, yield is 79%, GC content is 99%.
Embodiment 3
[0038] Example 3: Preparation of acryloylmorpholine
[0039] In a four-necked flask equipped with a spherical condenser and stirrer, add 1g p-hydroxyanisole, 21.6g (0.3mol) acrylic acid and 8.3g (0.06mol) phosphorus trichloride, and add 50ml of dichloromethane as a solvent , Lower the temperature to 0°C, add 57.4g (0.66mol) of morpholine (previously dissolved in 30ml of dichloromethane) into the reaction solution, slowly add dropwise, control the reaction temperature at 0~5°C, and finish the dropwise addition in 3.5 hours. Incubate the reaction for 1 hour, filter, and spin-dry the solvent to obtain 38 g of crude product, with a GC analysis content of 92%, and vacuum distillation to obtain 33.6 g, with a yield of 80% and a GC content of 99%.
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