Drying device
A drying device and drying technology, applied in the direction of drying gas arrangement, drying solid materials, drying, etc., can solve the problems of cumbersome process operation, high device requirements, and inability to fully meet industrial production, and achieve good dissolution rate and stability Good results
- Summary
- Abstract
- Description
- Claims
- Application Information
AI Technical Summary
Problems solved by technology
Method used
Image
Examples
Embodiment 1
[0044] Refer to the method reported in WO2012146099 and other literatures to prepare crude caspofungin acetate. Dissolve the crude product in ethanol solvent at a temperature of 15-20℃, maintain the temperature and filter the aforementioned solution into a fine drying bag, and gradually add ethyl acetate , Stir to crystallize, and filter to obtain a solid. Then carry out drying treatment as follows:
[0045] 1) Turn on the temperature control device, and the cooling liquid enters the gap between the inner and outer walls of the box (31) through the liquid inlet (315) provided on the box (31), so as to control the temperature in the drying device at -30~ -20℃ requirement;
[0046] 2) Open the box cover (32), place the sample of caspofungin acetate to be dried in the box body (31), close the box cover (32), close the pressure reducing valve, and use the vacuum device to dry the sample from the air outlet (5) Pump the vacuum carrier into the device and close the air outlet (5);
[00...
Embodiment 2
[0069] Example 2: Preparation of caspofungin with reference to literature methods
[0070] Caspofungin was prepared with reference to the method reported in WO2012146099, and the purity of caspofungin acetate to be dried was about 99.10%, and then passed through WO94 / 21677, WO2010008496, WO2009151341, J.Org.Chem., 2007,72,2335-2343, respectively. And the method of WO2010108637 to dry the obtained caspofungin acetate.
[0071] Sample solubility test
[0072] Take the aforementioned appropriate amount of caspofungin to be easily soluble in 0.1 mol / L hydrochloric acid and water, and dissolve in ethanol.
[0073] Inspection method: Method for determination of solubility in the second part of the Chinese Pharmacopoeia 2010
[0074] Operation method: Weigh the test sample, stir and dissolve it in a certain amount of solvent at 25℃±2℃. If there are no visible solute particles, it is regarded as completely dissolved.
[0075] According to relevant regulations of Chinese Pharmacopoeia: Solubilit...
PUM
Login to View More Abstract
Description
Claims
Application Information
Login to View More 


