Use of columbin, isocolumbin, deoxidized fibraurin in preparing antiphlogistic, stomach convulsion, stomach ache medicine
A technology of oxystigmata and bittern, which is applied in the field of medicine, can solve the problems of differences in cure rate and effective rate, no quality standards, and insufficient pharmacological screening, etc.
- Summary
- Abstract
- Description
- Claims
- Application Information
AI Technical Summary
Problems solved by technology
Method used
Image
Examples
Embodiment 1
[0132] Extract 2.5kg of dried medicinal material of Lavenderia quinquefolium, extract twice with 50 liters of 95% solution, 2 hours each time, combine the two extracts, concentrate under reduced pressure to obtain 120g of extract, disperse with 2 liters of water, and extract three times with 6L chloroform Concentrate the extraction part under reduced pressure to obtain 20 g of the crude product, heat and dissolve the crude product with 500 ml of methanol, filter while it is hot, and refrigerate the filtrate in a refrigerator at 4°C overnight to separate out the combination of columbin, isocolumbin and deoxyaldopicrin The product crystallized, filtered through filter paper, and dried to obtain 12g of the composition. Take 10g of the composition, mix it with 50g of silica gel as a sample, add it to the top of the silica gel column that has been installed, and use petroleum ether:chloroform (20:1~5:1) system Gradient elution, TLC tracking, combined eluents containing the same comp...
Embodiment 2
[0134] Tablet: active ingredient (three monomers or combination) 17g
[0135] Lactose 200g
[0136] Cornstarch 50g
[0138] Made into 1000 pieces
[0139] Preparation method: mix the active ingredient, lactose and starch, uniformly moisten with water to make a soft material, granulate the wetted mixture, pass through a 20-mesh sieve, dry at 80°C, add magnesium stearate, sieve again, and then The mixture is compressed into tablets, each tablet weighs 270 mg, and the active ingredient content is 17 mg.
[0140] The active ingredient of the present invention is combined with related carriers, and can also be made into other solid preparations, such as powders, granules, capsules and the like. The technology of these preparations is very mature, so I won't list them one by one here.
Embodiment 3
[0142] Infusion solution: active ingredient (three monomers or combination) 2g
[0144] Water for injection 100000ml
[0145] Makes 1000 bottles
[0146] Preparation method: Dissolve the active ingredient and sodium chloride in 100,000ml of water for injection, add 0.01% activated carbon for adsorption, detect intermediates, filter through a 0.45um membrane, subpackage, 100ml / bottle, sterilize, and inspect.
[0147] The active ingredients of the present invention can be combined with related adjuvants to make other liquid preparations, such as nasal sprays, injections and the like.
[0148] The above-mentioned pharmaceutical dosage forms can be effectively used for the treatment and prevention of acute and chronic inflammation, stomach spasm, stomach disease and related diseases.
PUM
Login to View More Abstract
Description
Claims
Application Information
Login to View More 