Method for preparing divinyl dipyridine compounds
A divinyl and bipyridine technology, applied in the field of preparation of divinyl bipyridine compounds, can solve the problems of low yield and short synthesis route, achieve good yield, easy separation, and avoid the use of highly toxic and dangerous drugs. effect used
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Embodiment 1
[0011] (1) Synthesis of 4,4'-dibromomethyl-2,2'-bipyridyl: in 300 milliliters of carbon tetrachloride, add 8 grams of 4,4'-dimethyl-2,2'-bipyridine Pyridine with 24 grams of N-bromosuccinimide (NBS), and 1 gram of azobisisobutyronitrile. Heated to reflux for 3 hours, cooled with ice water, and filtered to remove insoluble matter. The solvent was spun off to obtain light brown product 4,4'-dibromomethyl-2,2'-bipyridine 5.2 grams, yield 35%
[0012] (2) Synthesis of 4,4'-bis(diethylmethylphosphite)-2,2'-bipyridine (Wittig-Horner reagent): 6.8 grams of 4,4'-dibromomethyl-2 , 2'-bipyridyl and 60ml triethyl phosphite were mixed and stirred, refluxed for 4.5 hours and then cooled to room temperature. The unreacted triethyl phosphite was distilled off under reduced pressure, and the residue was refrigerated for 1 hour and then taken out, solidified into a dark brown solid, washed with 100 ml of ether, and dried under vacuum at 50 degrees Celsius to obtain 4,4'-bis( Diethylmethylph...
Embodiment 2
[0015] (1) Synthesis of 4,4'-dibromomethyl-2,2'-bipyridyl: in 400 milliliters of carbon tetrachloride, add 18.4 grams of 4,4'-dimethyl-2,2'-bipyridine Pyridine with 48 grams of N-bromosuccinimide (NBS), and 1 gram of azobisisobutyronitrile. Heated to reflux for 8 hours, cooled with ice water, and filtered to remove insoluble matter. The solvent was spun off to obtain brown product 4,4'-dibromomethyl-2,2'-bipyridine 12.6 grams, yield 37%
[0016] (2) Synthesis of 4,4'-bis(diethylmethylphosphite)-2,2'-bipyridine (Wittig-Horner reagent): 17.1 grams of 4,4'-dibromomethyl-2 , 2'-bipyridine was stirred with 90 ml of triethyl phosphite, heated to reflux, cooled to room temperature after 8 hours of reaction, unreacted triethyl phosphite was distilled off under reduced pressure, and the residue was placed in the refrigerator for 1 hour , solidified as a dark brown solid, washed with 150 milliliters of ether, and dried under vacuum at 50 degrees Celsius to obtain 19.4 grams of 4,4'-bi...
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