Pingyangmycin local injection preparation and preparation method thereof
A technology of local injection and pingyangmycin, which is used in pharmaceutical formulations, medical preparations with non-active ingredients, and drug delivery. effect, low viscosity
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Embodiment 1
[0022] A local injection preparation of pingyangmycin, comprising 0.05g of pingyangmycin hydrochloride, 2ml of absolute ethanol, 15g of soybean lecithin, 20g of glyceryl dioleate and 2g of poloxamer 407. The preparation method is as follows: first mix 0.05g of pingyangmycin hydrochloride with 2ml of absolute ethanol to form a suspension, then mix it with 15g of soybean lecithin, 20g of glyceryl dioleate and 2g of poloxamer 407, and keep stirring for 2h , and finally sterilized by filtration to obtain Pingyangmycin local injection preparation A1.
Embodiment 2
[0024] A local injection preparation of pingyangmycin, comprising 0.08g of pingyangmycin hydrochloride, 4ml of absolute ethanol, 20g of soybean lecithin, 25g of glyceryl dioleate and 2g of polyethylene glycol 200. The preparation method is as follows: first mix 0.08g of pingyangmycin hydrochloride with 4ml of absolute ethanol to form a suspension, then mix it with 20g of soybean lecithin, 25g of glyceryl dioleate and 2g of polyethylene glycol 200, and keep stirring for 3h , and finally sterilized by filtration to obtain Pingyangmycin local injection preparation A2.
Embodiment 3
[0026] A pingyangmycin local injection preparation, comprising 0.06g pingyangmycin hydrochloride, 3ml absolute ethanol, 20g egg yolk lecithin, 30g triolein and 3g poloxamer 407. The preparation method is as follows: mix 0.06g pingyangmycin hydrochloride, 20g egg yolk lecithin, 30g triolein and 3g poloxamer 407, keep stirring for 4 hours, and finally filter and sterilize to obtain pingyangmycin local injection preparation A3 .
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