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Nitrogen-containing heterocyclic derivative having 2-imino group and pest control agent including the same

A pest control, imino technology, applied in biocides, insecticides, animal repellents, etc., can solve the problems of drug sensitivity and safety reduction

Pending Publication Date: 2019-09-20
MMAG CO LTD
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0021] The present invention is designed to provide a new pest control agent in order to solve problems in the field of pest control such as reduction of drug susceptibility, long-term effect, safety in use, etc.

Method used

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  • Nitrogen-containing heterocyclic derivative having 2-imino group and pest control agent including the same
  • Nitrogen-containing heterocyclic derivative having 2-imino group and pest control agent including the same
  • Nitrogen-containing heterocyclic derivative having 2-imino group and pest control agent including the same

Examples

Experimental program
Comparison scheme
Effect test

Embodiment

[0868] Next, the present invention is described more specifically with reference to Examples, but the present invention is not limited to the Examples.

[0869] Reference Example 1: N-[1-((6-chloropyridin-3-yl)methyl)pyridin-2(1H)-ylidene]-2,2,2-trifluoroacetamide (compound P212)

[0870] (1) 25 g (270 mmol) of 2-aminopyridine was dissolved in 200 mL of anhydrous dichloromethane, 41 mL (30 g, 300 mmol) of triethylamine was added, and the mixture was cooled to 0°C. 38 mL (57 g, 270 mmol) of anhydrous trifluoroacetic acid was added dropwise over 15 minutes, and the resulting mixture was stirred at room temperature for 2 hours. After the reaction was completed, the reaction solution was poured into about 100 mL of ice water, and the mixture was stirred for 10 minutes. The mixture was moved to a separatory funnel for liquid separation, and the organic layer was washed twice with 150 mL of water and twice with 150 mL of 1% aqueous HCl, dried over anhydrous magnesium sulfate, and c...

preparation Embodiment 1

[1191] Preparation Example 1 [Granules]

[1192]

[1193] The above ingredients are uniformly ground and mixed, water is added to knead the ingredients well, and the mixture is then granulated and dried to obtain granules.

preparation Embodiment 2

[1194] Preparation Example 2 [Granules]

[1195]

[1196] The above ingredients are uniformly ground and mixed, water is added to knead the ingredients well, and the mixture is then granulated and dried to obtain granules.

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PUM

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Abstract

Provided is a nitrogen-containing heterocyclic derivative having a 2-imino group, which is represented by the following Formula (I). [in the formula, Ar represents a phenyl group which may be substituted, a 5- to 6-membered heterocycle which may be substituted, or a 4- to 10-membered heterocycloalkyl group, A represents a heterocycle having a 5- to 10-membered unsaturated bond including one or more nitrogen atoms, and has an imino group substituted with an R group at a position adjacent to the nitrogen atom present on the cycle, Y represents a hydrogen atom, a halogen atom, a hydroxyl group, a C1 to C6 alkyl group which may be substituted with a halogen atom, a C1 to C6 alkyloxy group which may be substituted with a halogen atom, a cyano group, or a nitro group, and R represents any one of groups represented by the following Formulae (a) to (e), (y) or (z).].

Description

[0001] This application is a divisional application of PCT application PCT / JP2013 / 056055, which was submitted on February 27, 2013 and has an invention title of "Nitrogen-containing heterocyclic derivatives having 2-imino groups and pest control agents containing the same". The date when the above-mentioned PCT application entered the national phase in China was September 10, 2014, and the application number was 201380013407.1. [0002] [Technical field] [0003] The present invention relates to a nitrogen-containing heterocyclic derivative having a 2-imino group and a new pest control agent using the same. [0004] [Background technique] [0005] Although many pest control agents have been discovered so far, new drugs are still needed due to problems such as reduced drug sensitivity, long-term effects, and safety during use. [0006] Especially for rice cultivation in East and Southeast Asia, damage caused by planthoppers that have developed resistance to major insecticides c...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): C07D213/74C07D401/06C07D405/06C07D417/06C07D213/75C07F9/58A01N43/40A01N43/78A01N43/60A01N43/58A01N43/54A01N43/76A01P7/04
CPCA01N43/40A01N43/54A01N43/78A01N57/32C07D213/75C07D401/06C07D405/06C07D417/06C07F9/58C07D213/74A61P33/00
Inventor 利部伸三三富正明橘田繁辉堀越亮小野崎保道中村哲
Owner MMAG CO LTD
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