A kind of synthetic method of m-aminoacetanilide hydrochloride
A technology of aminoacetanilide hydrochloride and synthesis method, which is applied in the field of synthesis of m-aminoacetanilide hydrochloride, can solve the problems of high energy consumption, long reaction cycle, high reaction temperature, etc., and achieve high yield and product yield High, easy-to-operate effect
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Embodiment 1
[0025] Stir and add 150g of 50% acetic acid into a 500ml four-necked bottle, stir and add 54.0g of m-phenylenediamine, and add 59.88g of hydrochloric acid (32%) dropwise at 15-25°C for 30 minutes, stir until the material dissolves, and then cool down in an ice bath to 0-25°C. 5°C. Add 53.6g of acetic anhydride at 0~5°C over 4~5h. After the addition, the reaction was continued at this temperature for 1 hour, and sampling was carried out. The raw materials were 0.71%, m-aminoacetanilide hydrochloride 90.2%, m-diacetanilide hydrochloride 8.04%, filtered to obtain m-aminoacetanilide hydrochloride wet cake 96.3g , purity 98.91%, amino value 84.57%, yield 88.21%, mother liquor 205.3g (raw material 14.23%, m-aminoacetanilide hydrochloride 35.76%, m-diacetanilide 47.5%) is used in the next batch.
Embodiment 2
[0027] Add 150 g of the mother liquor in Example 1 into the flask, add 59.88 g of hydrochloric acid (32%), stir and heat up to 80° C. Insulate at 80-90°C for 1h. Cool down to 60°C, take samples to detect the content of hydrochloric acid and acetic acid, the content of hydrochloric acid is 10.4%, and the content of acetic acid is 40.1%. Add 54g of m-phenylenediamine, stir to dissolve, and lower the temperature to 0-5°C at the same time. Add 58.3g of acetic anhydride dropwise over 4 to 5 hours, and keep warm at 0 to 5°C for 1 hour after the addition, and detect that the raw material is 0.32%, m-aminoacetanilide hydrochloride is 91.61%, and m-diacetanilide is 7.84%. After the end point, filter to obtain m-aminoacetanilide hydrochloride wet cake 107.5g, purity 99.0%, amino value 84.25%, yield 98.10%, mother liquor 190.2g (raw material 15.65%, m-aminoacetanilide hydrochloride 37.16%, Between diacetamidoaniline 46.22%) cover for next batch.
Embodiment 3
[0029] Add 150 g of the mother liquor in Example 2 into the flask, add 59.88 g of hydrochloric acid (32%), stir and heat up to 80° C. Insulate at 80-90°C for 1h. Cool down to 60°C, take samples to detect the content of hydrochloric acid and acetic acid, the content of hydrochloric acid is 10.7%, and the content of acetic acid is 39.5%. Add 54g of m-phenylenediamine, stir to dissolve, and lower the temperature to 0-5°C at the same time. Add 58.3g of acetic anhydride dropwise over 4 to 5 hours, and keep warm at 0 to 5°C for 1 hour after the addition, and detect that the raw material is 0.51%, m-aminoacetanilide hydrochloride is 90.47%, and m-diacetanilide is 8.52%. After the end point, filter to obtain 107.7g of m-aminoacetanilide hydrochloride wet cake, with a purity of 98.93%, an amino value of 84.42%, and a yield of 98.48%. The mother liquor 187.1g is used in the next batch.
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