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Process for preparing sulodexide raw material

A preparation process and process technology, applied in the field of sulodexide raw material production, can solve the problems affecting the extraction of sulodexide substances, low purity of sulodexide raw materials, unsuitable for industrialized production, etc. Amplified, practical effect

Inactive Publication Date: 2021-12-03
江苏唯高生物科技有限公司
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0004] The purpose of the present invention is to provide a process for preparing sulodexide raw material, so as to solve the problem that the existing process for preparing sulodexide raw material proposed in the above background technology is easy to introduce impurities, complex process, high cost, and is not suitable for industrial production. , and the purity of the prepared sulodexide raw material is not high, which affects the extraction of sulodexide substances

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0025] A kind of technique for preparing sulodexide raw material, concrete preparation process steps are as follows:

[0026] Step 1: adding chondroitin sulfate, dermatan sulfate, nucleic acid and heparin sodium to the mixed solution of heparin sodium to better separate heparin sodium from impurities, and collecting the precipitate to obtain a crude heparin sodium solution;

[0027] Step 2: under low temperature conditions, adjust the pH value of the crude heparin sodium aqueous solution to acidity, centrifuge at low temperature, and collect the supernatant to obtain a sulfated polysaccharide solution;

[0028] Step 3: Add 1 kg of sulfated polysaccharide solution, add water to dissolve to 5-15% mmol / L, add calcium chloride to make the concentration 1-10 mmol / L (preferably 4 mmol / L), add magnesium sulfate to make the magnesium ion concentration 1-10 mmol / L L (preferably 2-5mmol / L), add sodium chloride to make the concentration 0.1%~1.5%mmol / L (preferably 0.3-0.5%mmol / L), use el...

Embodiment 2

[0040] A kind of technique for preparing sulodexide raw material, concrete preparation process steps are as follows:

[0041] Step 1: adding chondroitin sulfate, dermatan sulfate, nucleic acid and heparin sodium to the mixed solution of heparin sodium to better separate heparin sodium from impurities, and collecting the precipitate to obtain a crude heparin sodium solution;

[0042] Step 2: under low temperature conditions, adjust the pH value of the crude heparin sodium aqueous solution to acidity, centrifuge at low temperature, and collect the supernatant to obtain a sulfated polysaccharide solution;

[0043] Step 3: 1 kg of sulfated polysaccharide solution, add water to dissolve to 5-15% mmol / L, add sodium chloride to make the concentration 1-10 mmol / L (preferably 4 mmol / L), add magnesium sulfate to make the magnesium ion concentration 1-10 mmol / L L (preferably 2-5mmol / L), add sodium chloride to make the concentration 0.1%~1.5%mmol / L (preferably 0.3-0.5%mmol / L), use electri...

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PUM

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Abstract

The invention discloses a process for preparing a sulodexide raw material, the process comprises the following specific preparation process steps: step 1, adding chondroitin sulfate, dermatan sulfate, nucleic acid and heparin sodium into a heparin sodium mixed solution to better separate heparin sodium from impurities, and collecting precipitate to obtain a crude heparin sodium solution; step 2, under the low-temperature condition, adjusting the pH value of the heparin sodium crude product water solution to be acidic, performing low-temperature centrifugation, collecting supernate, and obtaining a sulfated polysaccharide solution; and step 3, adding water into 1kg of sulfated polysaccharide solution to dissolve the sulfated polysaccharide solution until the concentration is 5-15% mmol / L, adding calcium chloride until the concentration is 1-10mmol / L (preferably 4mmol / L), adding magnesium sulfate until the concentration of magnesium ions is 1-10mmol / L (preferably 2-5mmol / L), and adding sodium chloride until the concentration is 0.1-1.5% mmol / L (preferably 0.3-0.5% mmol / L). The process for preparing the sulodexide raw material is stable and reliable, simple in equipment, convenient to operate, high in practicability and suitable for being widely popularized and used.

Description

technical field [0001] The invention belongs to the technical field of sulodexide raw material production, and in particular relates to a process for preparing sulodexide raw material. Background technique [0002] Sulodexide was first developed by the Italian Alpha Wessman Pharmaceutical Company and was launched in 1974. It is extracted and refined from pig intestinal mucosa. It is a highly purified glycosaminoglycan, belonging to heparinoids, and its chemical composition is 80% fast-moving heparin. Sulodide has been used as an antithrombotic drug to treat various cardiovascular diseases for more than 20 years. It is currently used as an antithrombotic drug to treat peripheral cardiovascular diseases in Italy, Spain, Eastern Europe, South America and Asia. It was introduced in my country in the 1990s Start importing. [0003] Compared with heparin, sulodexide has stronger antithrombotic potential under the premise of reducing bleeding, and has a longer half-life, and lower...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): C08B37/10
CPCC08B37/0075
Inventor 邱军捷
Owner 江苏唯高生物科技有限公司