Synthesis method of full halogenated miscellaneous naphthene
A technology of heterocycloalkane and synthesis method, which is applied in the field of synthesis of perhalogenated heterocycloalkane, and can solve problems such as high reaction temperature and harsh reaction conditions
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Embodiment 1
[0023] In a 1000ml four-neck flask with mechanical stirring and a reflux condenser, add 329g (1.0mol) of 1-bromo-2,2-diacetoxypentafluoropropane, 280g (2.0mol) of difluoromalonic acid, 10g of para Toluenesulfonic acid, stirred, heated to 120 ° C, regularly sampled and analyzed, when it was detected that the reaction was over, cooled, and 272g of 2-trifluoromethyl-2-difluorobromomethyl-4,6-dioxo-5 was isolated -Difluoro-1,3-dioxane, yield 78%.
[0024] In a 1000ml pressure reactor, add 175g (0.5mol) of the above-prepared 2-trifluoromethyl-2-difluorobromomethyl-4,6-dioxo-5-difluoro-1,3-diox Heterocyclohexane, 300g dichloromethane, 324g sulfur tetrafluoride, stirred, and reacted at 120°C. After the reaction, cooled and separated to obtain 106g 2-trifluoromethyl-2-difluorobromomethyl-4 , 4,6,6-tetrafluoro-5-difluoro-1,3-dioxane, the yield was 54%, and the corresponding hydrogen-containing dioxane impurity was not detected.
Embodiment 2
[0026] In a 500ml four-neck flask with mechanical stirring and reflux condenser, add 268g (1.0mol) 2,2-diacetoxyhexafluoropropane, 108g oxalic acid (1.2mol), 5g concentrated sulfuric acid, stir, and heat up to 140°C , regular sampling analysis, when it is detected that the reaction is over, it is cooled to separate 201.5g2,2-bis(trifluoromethyl)-4,5-dioxo-1,3-dioxolane, yield 84.7%.
[0027]In a 1000ml four-neck flask with mechanical stirring and a reflux condenser, add 312g (1.5mol) of phosphorus pentachloride, 500g of phosphorus oxychloride and 119g (0.5mol) of the 2,2-bis(trifluoromethyl) prepared above )-4,5-dioxo-1,3-dioxolane, stirred, heated to 100°C, and reacted at 100°C. After the reaction, 142g of 2,2-bis(trifluoromethyl)-4,4,5,5-tetrachloro-1,3-dioxolane was separated by cooling, the yield was 81.6%, and no corresponding Hydrogen-containing dioxolane impurity.
Embodiment 3
[0029] In a 1000ml four-neck flask with mechanical stirring and reflux condenser, add 301g (1.0mol) 1,3-dichloro-2,2-diacetoxytetrafluoropropane, 180g (2mol) oxalic acid, 30g trichloride Iron, 300g of 1-ethyl-3-methylimidazolium tetrafluoroborate, stirred, heated up to 50°C, regularly sampled and analyzed, when it was detected that the reaction was over, cooled, and 250.7g of 2,2-bis(difluorochloro Methyl)-4,5-dioxo-1,3-dioxolane, yield 92.5%.
[0030] In a 1000ml four-neck flask with mechanical stirring and a reflux condenser, add 136g (0.5mol) of 2,2-bis(difluorochloromethyl)-4,5-dioxo-1,3- Dioxolane, 100g DMF, stirred, heated up to 70°C, 357g (3.0mol) of thionyl chloride was added dropwise, and after the addition of thionyl chloride was completed, the reaction was carried out under reflux. After the reaction was completed, 85.5g of 2,2-bis(difluorochloromethyl)-4,4,5,5-tetrachloro-1,3-dioxolane was obtained by cooling and separation, with a yield of 45%, undetected Out of...
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