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A preparing method of a radix notoginseng total saponin transdermal agent

The technology of total saponins of Panax notoginseng and transdermal agent is applied in the field of preparation of transdermal agent, which can solve the problems of inconvenient clinical administration of liquid preparations, limited utilization and the like, and achieves the effects of improving immunity of the body, relieving local symptoms, and quick effect.

Inactive Publication Date: 2016-10-19
TIANJIN PHARMACN MEDICAL TECH
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

However, when it is used as a topical preparation, it is often limited due to the inconvenience of clinical administration of liquid preparations.

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0028] A panax notoginseng total saponin transdermal agent mainly contains notoginseng total saponin, and the encapsulation rate is 86.79±1.68%.

[0029] The preparation method of the aforementioned panax notoginseng saponins transdermal agent, the specific preparation steps are as follows:

[0030] (1) The total saponins of Panax notoginseng are superfinely crushed and passed through a 200-mesh sieve;

[0031] (2) Weigh 25g of panax notoginseng saponins as raw materials;

[0032] (3) Add the panax notoginseng saponins to 1L of absolute ethanol, magnetically stir for 6 hours in a sealed explosion-proof environment at room temperature;

[0033] (4) Put the solution obtained in step (3) into distilled water with a V / V of 16:1, stir for 30 minutes, and set aside;

[0034] (5) Dissolve 1 g of chitosan in 32 mL of 1% glacial acetic acid solution, stir and dissolve the chitosan glacial acetic acid solution, where the stirring temperature is 45-55°C, and the heating method is steam heating;

[0...

Embodiment 2

[0044] A panax notoginseng total saponin transdermal agent mainly contains notoginseng total saponin, and the encapsulation rate is 84.89±1.79%.

[0045] The preparation method of the aforementioned panax notoginseng saponins transdermal agent, the specific preparation steps are as follows:

[0046] (1) The total saponins of Panax notoginseng are superfinely pulverized and passed through a 300-mesh sieve;

[0047] (2) Weigh 30g of panax notoginseng saponins as raw materials;

[0048] (3) Add the panax notoginseng saponins to 1L of absolute ethanol, magnetically stir for 6 hours in a sealed explosion-proof environment at room temperature;

[0049] (4) Put the solution obtained in step (3) into distilled water with a V / V of 16:1, stir for 30 minutes, and set aside;

[0050] (5) Dissolve 7.5 g of chitosan in 160 mL of 2% glacial acetic acid, stir to dissolve the chitosan glacial acetic acid solution, the stirring temperature is 45° C., and the heating method is steam heating.

[0051] (6) Di...

Embodiment 3

[0060] A panax notoginseng total saponin transdermal agent mainly contains notoginseng total saponin, and the encapsulation rate is 81.89±1.33%.

[0061] The preparation method of the aforementioned panax notoginseng saponins transdermal agent, the specific preparation steps are as follows:

[0062] (1) The total saponins of Panax notoginseng are superfinely crushed and passed through a 100-mesh sieve;

[0063] (2) Weigh 28g of panax notoginseng saponins as raw materials;

[0064] (3) Add the panax notoginseng saponins to 1L of absolute ethanol, magnetically stir for 6 hours in a sealed explosion-proof environment at room temperature;

[0065] (4) Put the solution obtained in step (3) into distilled water with a V / V of 16:1, stir for 30 minutes, and set aside;

[0066] (5) Dissolve 1.8 g of chitosan in 32 mL of 3% glacial acetic acid, stir to dissolve the chitosan glacial acetic acid solution, the stirring temperature is 55° C., and the heating method is steam heating.

[0067] (6) Dissol...

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Abstract

A preparing method of a radix notoginseng saponin transdermal agent is disclosed. The method includes steps of (1) dissolving radix notoginseng saponins into absolute alcohol and distilled water in order, (2) heating to prepare a chitosan-glacial acetic acid solution, (3) mixing a traditional Chinese medicine extract liquid with the chitosan-glacial acetic acid solution, (4) adding the mixture into an emulsification system, and emulsifying, (5) crosslinking emulsified products, and (6) treating a product of the crosslinking reaction through washing, precipitating, centrifuging and drying to obtain a transdermal medical membrane loaded with the traditional Chinese medicine extract liquid. The method is simple and suitable for needs of large-scale industrial production.

Description

Technical field [0001] The invention relates to a preparation method of a transdermal agent, in particular to a preparation method of a panax notoginseng saponins transdermal agent. Background technique [0002] Panax notoginseng saponins are the main active alkaloids in the traditional Chinese medicine Panax notoginseng. Modern medical research shows that Panax notoginseng saponins have various effects such as dilating blood vessels, preventing thrombosis, inhibiting platelet aggregation, and improving cerebral ischemia. They are widely used in clinical practice. For the treatment of ischemic cerebrovascular disease and achieve a relatively ideal therapeutic effect, according to the results of pharmacokinetics, Panax notoginseng saponins have the characteristics of fast absorption, fast metabolism, and short half-life (2.8 hours). In the injection mode, frequent administration is required to maintain the effective blood concentration of the drug, so it is necessary to develop it...

Claims

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Application Information

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IPC IPC(8): A61K9/70A61K36/258A61K47/36A61P9/10
Inventor 田东奎何磊
Owner TIANJIN PHARMACN MEDICAL TECH