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Method for preparing sn-1-DHA-hemolytic phosphatidylserine

A technology of phosphatidylserine and glycerophosphorylserine is applied in the field of preparing sn-1-DHA-lysophosphatidylserine, which can solve the problems of reducing the utilization efficiency of DHA and the transportation efficiency, and achieve the effect of high DHA purity

Active Publication Date: 2019-06-07
威海深蓝奇迹生物科技有限公司
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0004] DHA lysophosphatidylserine is usually divided into sn-1-DHA-lysophosphatidylserine and sn-2-DHA-lysophosphatidylserine according to the different positions of DHA on the glycerol backbone, and the DHA in the latter will be due to The action of phospholipase A2 in the human body produces free DHA and glycerol phosphatidylserine, which reduces the utilization efficiency of DHA and the delivery efficiency to the brain to a certain extent. Therefore, sn-1-DHA-lysophosphatidylserine is DHA lysophospholipid A better chemical form of acylserine, but there is currently no mature preparation method for this product

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0040] A method for preparing sn-1-DHA-lysophosphatidylserine, comprising the following steps:

[0041] (1) Weigh 5.0g of soybean phosphatidylserine (wherein phosphatidylserine accounts for 35% of the total phospholipids) and dissolve it in 20mL of n-hexane, add 15g of absolute ethanol and 1.5g of immobilized Candida antarctica lipase Lipozyme 435 (provided by Novozymes), heated to 60 ° C and stirred for 2 h, then filtered the reaction mixture to reclaim the immobilized Candida antarctica enzyme, and the filtrate was removed at 60 ° C and -0.088 MPa to remove n-hexane solvent and unreacted ethanol. Then add 50mL of acetone to fully shake and wash and collect the acetone insoluble matter;

[0042] (2) Dissolve the acetone-insoluble material obtained in step (1) in 20 mL of chloroform after evaporating to dry acetone, add 1.0 g of absolute ethanol and 1.5 g of Lipozyme 435, stir and react at 60°C for 8 hours, then keep 60°C and apply Vacuum to remove chloroform solvent and unre...

Embodiment 2

[0045] (1) Weigh 5.0g of soybean phosphatidylserine (wherein phosphatidylserine accounts for 50% of the total phospholipids) and dissolve it in 20mL of n-hexane, add 5.0g of absolute ethanol and 0.05g of immobilized Candida antarctica lipase Lipozyme 435 and heat Stir the reaction at 30°C for 8 hours, then filter the reaction mixture to recover the immobilized enzyme, remove the n-hexane solvent and unreacted ethanol from the filtrate at 60°C and -0.088MPa, then add 50mL of acetone to fully shake and wash, and collect the acetone insoluble matter;

[0046] (2) Dissolve the acetone-insoluble material obtained in step (1) in 20 mL of chloroform after evaporating the acetone, add 0.5 g of absolute ethanol and 0.05 g of Lipozyme 435, stir and react at 30 ° C for 24 h, then heat to 60 ° C and add to the reaction Vacuum was applied to the system to remove chloroform solvent and unreacted ethanol, then 10 mL of deionized water was added and stirred thoroughly, then suction filtered, t...

Embodiment 3

[0049] (1) Weigh 5.0 g of soybean phosphatidylserine (wherein phosphatidylserine accounts for 80% of the total phospholipids) and dissolve it in 20 mL of n-hexane, add 10 g of absolute ethanol and 0.5 g of immobilized Candida antarctica lipase Lipozyme 435 and heat for 40 Stir the reaction at ℃ for 2 hours, then filter the reaction mixture to recover the immobilized enzyme, remove the n-hexane solvent and unreacted ethanol from the filtrate under the condition of 60 ℃ and -0.088MPa, then add 50mL acetone to fully shake and wash, and collect the acetone insoluble matter;

[0050] (2) Dissolve the acetone-insoluble material obtained in step (1) in 20 mL of chloroform after evaporating the acetone, add 0.5 g of absolute ethanol and 0.05 g of Lipozyme 435, stir and react at 30°C for 24 hours, then heat to 60°C and apply Vacuum to remove chloroform solvent and unreacted ethanol, then add 10mL deionized water and stir well, then filter with suction, then centrifuge the filtrate, disc...

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Abstract

The invention relates to the technical field of health-care food, in particular to a method for preparing sn-1-DHA-hemolytic phosphatidylserine. The method comprises the following steps: carrying outalcoholysis on phosphatidylserine to obtain glycerol phosphorylserine, and then carrying out ester synthesis reaction with DHA. The method for preparing sn-1-DHA-hemolytic phosphatidylserine preparesthe high-purity sn-1-DHA-hemolytic phosphatidylserine through two steps of alcoholysis and one step of ester synthesis reaction.

Description

technical field [0001] The invention relates to the technical field of health food, in particular to a method for preparing sn-1-DHA-lysophosphatidylserine. Background technique [0002] Marine animal phospholipids are a class of phospholipids derived from marine animal tissues and rich in omega-3 fatty acids such as docosahexaenoic acid (DHA) and eicosapentaenoic acid (EPA). Different from traditional DHA products such as fish oil and algae oil DHA, DHA and phospholipids in DHA phospholipids are combined by chemical bonds. In addition to having the dual physiological functions of DHA and phospholipids, it also plays a synergistic effect of "1+1>2" , known as "the latest generation of DHA products". The human cell membrane structure is a typical phospholipid bilayer structure. The chemical structure of DHA phospholipids makes it have a higher affinity with human cells, tissues and organs, and the digestion and absorption rate of DHA phospholipids in the human body is clo...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): C12P13/06C12P7/64
Inventor 蔡胜利孙兆敏蔡爱英曾海亭
Owner 威海深蓝奇迹生物科技有限公司