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Application of elaeocarpus nitentifolius extract in preparation of medicines for treating stomach-related diseases

A technology of extracts and medicines, applied in the field of medicine, can solve problems such as the lack of reports on the research on the treatment of stomach diseases by Du Ying with bright leaves

Active Publication Date: 2021-05-28
INST OF MATERIA MEDICA AN INST OF THE CHINESE ACAD OF MEDICAL SCI
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0003] In a large number of screening work, we found that the extract of Du Ying has a high gastric H + -K + -ATPase inhibitory activity, the extract has a significant protective effect on gastric mucosal bleeding caused by indomethacin and cold stress, so far there is no report on the treatment of gastric diseases by Liangye Duying

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0017] The preparation (water extraction extract) of embodiment 1 bright leaf Du Ying extract

[0018] 1 kg of the branches and leaves of Du Ying with distilled water were extracted three times under hot reflux with distilled water, each time for one hour, and the extract was concentrated under reduced pressure to obtain 70 g of water extract.

Embodiment 2

[0019] The preparation of embodiment 2 Du Ying radix extract (example of alcohol extraction extract)

[0020] 2.2 kg of Du Ying leaves, add 6 times the amount of 90% ethanol, soak overnight or 4 hours, slowly heat to boiling, reflux for 1 hour, filter; repeat the whole process twice, combine the filtrate, concentrate under reduced pressure, temperature 60-70 ℃, Pressure 85-98KPa, when concentrated to completely free of ethanol, add water of the same weight as the medicinal materials and continue heating until boiling, after cooling, centrifuge to remove insoluble matter, and add a small amount of water to wash the insoluble matter three times, combine the filtrates, and reduce pressure at a temperature of 60-70C Concentrate, then dry under reduced pressure (temperature 70-80°C, pressure 85-98Kpa) to obtain 147g of extract.

[0021] Pharmacological experiment:

[0022] The samples used in the pharmacological experiments are the samples obtained from the preparation of the extr...

experiment example 1

[0023] Experimental example 1. the extract of Duying radix L. to H + -K + -ATPase activity effect

[0024] Method: take a 96-well plate, add lysozyme, 1.0mg / ml and 0.25mg / ml of the extract of Duying radix, rabeprazole sodium 10 -3 mol / L and 10 -4 mol / L, the volume is 20ul. Add pig H diluted 20 times with the reaction solution + -K + -ATPase 160ul, incubate at 37°C for 20 minutes, add 20mg / ml ATP 20ul, blank without adding ATP. React at 37°C for 30 minutes. Add 50ul of 10% TCA to terminate the reaction. Blank plus 20mg / ml ATP20ul. Take 50 μl and place it in a 96-well microtiter plate, add 200ul of phosphorous solution for color reaction, and measure the color at 660nm. Calculate the inhibition rate, inhibition rate=(control-sample) / (control-blank)×100%.

[0025] RESULTS: The extract of Duying radix had a positive effect on pig stomach H + -K + -ATPase activity has a strong inhibitory effect, and the inhibition rates of 100ug / ml and 20ug / ml are 58% and 26%, respectiv...

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PUM

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Abstract

The invention discloses application of an elaeocarpus nitentifolius extract in preparation of an H<+>-K<+>-ATP enzyme inhibitor and an application of the elaeocarpus nitentifolius extract in preparation of medicines for preventing or treating stomach-related diseases. The invention further discloses a preparation method of the elaeocarpus nitentifolius extract. The stomach related diseases comprise gastric mucosa bleeding, gastric ulcer and reflux esophagitis. The gastric mucosa bleeding comprises gastric mucosa bleeding caused by anti-inflammatory pain and gastric mucosa bleeding caused by cold stress.

Description

technical field [0001] The present invention belongs to the technical field of medicine, and specifically relates to the new application of the extract of Duying radix, that is, the application of the extract of Duying liangye in the preparation of drugs for the prevention or treatment of stomach-related diseases, and in the preparation of H + -K + - Use in ATPase inhibitors. Background technique [0002] Elaeocarpus nitentifolius is a plant of the genus Elaeocarpus nitentifolius, about 200 species of which are distributed in East Asia, Southeast Asia, Southwest Pacific and Oceania. There are 38 species and 6 varieties in China, which are mainly distributed in South China and Southwest China. They are common middle-level trees in broad-leaved evergreen forests. Bright-leaved Duying is mainly produced in Guangdong, Guangxi, Vietnam and other places. It is a warm, neutral and partial shade tree species, and is mainly used as a beautiful garden ornamental tree species. No me...

Claims

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Application Information

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IPC IPC(8): A61K36/185A61P1/04A61P1/00A61P7/04
CPCA61K36/185A61P1/00A61P1/04A61P7/04A61K2236/331A61K2236/333
Inventor 康洁朱海波徐瑞明陈若芸杨柳王贵彬
Owner INST OF MATERIA MEDICA AN INST OF THE CHINESE ACAD OF MEDICAL SCI