Unlock instant, AI-driven research and patent intelligence for your innovation.

Preparation process of nanometer carboxymethyl chitosan particle as medicine carrier

A technology of carboxymethyl chitosan and nanoparticles, which can be used in pharmaceutical formulations, medical preparations of non-active ingredients, powder delivery, etc. It can solve the problems of large energy requirements and side effects of organic solvents, and meet environmental protection requirements , avoid side effects, process safety effect

Inactive Publication Date: 2008-06-04
WUHAN UNIV OF TECH
View PDF5 Cites 0 Cited by
  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0003] The existing preparation method of carboxymethyl chitosan nanoparticle adopts solvent evaporation and emulsification-solvent diffusion method, has adopted organic solvent, and organic solvent has side effect, and required energy is large

Method used

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
View more

Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0013] A kind of preparation method of drug carrier carboxymethyl chitosan nano particle, it comprises the steps:

[0014] 1). Dissolve carboxymethyl chitosan in distilled water at room temperature to obtain a carboxymethyl chitosan aqueous solution with a concentration of 0.5 mg / mL; 2). Add 0.1M carboxymethyl chitosan dropwise to the carboxymethyl chitosan aqueous solution The hydrochloric acid adjustment carboxymethyl chitosan aqueous solution pH value is 1, under stirring condition, adding concentration is 0.3mg / mL sodium tripolyphosphate aqueous solution, press carboxymethyl chitosan aqueous solution: sodium tripolyphosphate volume aqueous solution ratio= 1:1.5, adding sodium tripolyphosphate aqueous solution to obtain a mixture; 3). The obtained mixture was stirred until the cross-linking was complete, then centrifuged at a high speed, and freeze-dried to obtain drug carrier carboxymethyl chitosan nanoparticles with a particle size of 90-220nm .

[0015] When encapsulati...

Embodiment 2

[0017] A kind of preparation method of drug carrier carboxymethyl chitosan nano particle, it comprises the steps:

[0018] 1). Dissolve carboxymethyl chitosan in distilled water at room temperature to obtain a carboxymethyl chitosan aqueous solution with a concentration of 2.0mg / mL; 2). Add 0.1M carboxymethyl chitosan dropwise to the carboxymethyl chitosan aqueous solution sodium hydroxide to adjust the pH value of carboxymethyl chitosan aqueous solution to 6, and under stirring conditions, adding a concentration of 1.8 mg / mL calcium chloride aqueous solution, according to the volume ratio of carboxymethyl chitosan aqueous solution: calcium chloride aqueous solution =1:2.5, add calcium chloride aqueous solution to obtain the mixture; 3). The obtained mixture is stirred until the cross-linking is complete, high-speed centrifugation, freeze-drying to obtain drug carrier carboxymethyl chitosan nanoparticles with a particle size of 90-220nm .

[0019] When encapsulating the medic...

Embodiment 3

[0021] A preparation method of drug-loaded carboxymethyl chitosan nanoparticles, at room temperature, 40mg carboxymethyl chitosan is dissolved in 20mL distilled water, and the obtained concentration is 2.0mg / mL carboxymethyl chitosan aqueous solution; add 0.1M hydrochloric acid dropwise to the carboxymethyl chitosan aqueous solution to adjust the pH value of the carboxymethyl chitosan aqueous solution to be 2, then dissolve 10 mg of the model drug bovine serum albumin in the carboxymethyl chitosan solution, Serum albumin concentration was 0.5 mg / mL; then 4 mL of 1.4 mg / mL sodium tripolyphosphate aqueous solution was added to 2 mL of carboxymethyl chitosan solution to obtain a mixture; the mixture was stirred at room temperature until cross-linking was complete, then centrifuged at 12000rmp Separating and freeze-drying to obtain drug-loaded carboxymethyl chitosan nanoparticles with a particle diameter of 90-220 nm. The prepared nanoparticles are more regular spherical. The enc...

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
Login to View More

PUM

PropertyMeasurementUnit
particle diameteraaaaaaaaaa
concentrationaaaaaaaaaa
Login to View More

Abstract

The present invention relates to preparation process of nanometer carboxymethtyl chitosan particle as medicine carrier. The preparation process includes the following steps: 1. dissolving carboxymethtyl chitosan in water at room temperature to prepare 0.5-2.0 mg / mL concentration water solution of carboxymethtyl chitosan; 2. preparing mixture in one of two methods; and 3. stirring the mixture until complete cross-linking, high speed centrifugal separation and freeze drying to obtain the nanometer carboxymethtyl chitosan particle of size 90-220 nm for carrying medicine. The preparation process has mild condition and no side effect of organic solvent, and the nanometer carboxymethtyl chitosan particle is especially suitable for carrying sensitive macro molecule, such as protein matter.

Description

technical field [0001] The invention relates to a preparation method of drug carrier-carboxymethyl chitosan nanoparticles. Background technique [0002] Due to its high adhesion and good biocompatibility, chitosan has been widely used in drug carriers and medical auxiliary materials. Chitosan is insoluble in water when the pH value is above 6, which makes it not suitable for adsorbing ions under neutral conditions; after carboxymethylation, it inhibits the formation of hydrogen bonds between the amino groups and hydroxyl groups of chitosan, thereby improving water solubility. It has good water solubility under acid and alkali conditions. Carboxymethyl chitosan has polyviscosity, which can enhance the permeability and absorption of mucosal cells. [0003] The existing method for preparing carboxymethyl chitosan nanoparticles adopts solvent evaporation and emulsification-solvent diffusion methods, and uses organic solvents, which have side effects and require a lot of energy...

Claims

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
Login to View More

Application Information

Patent Timeline
no application Login to View More
Patent Type & Authority Patents(China)
IPC IPC(8): A61K47/36A61K9/14
Inventor 徐咏梅郑化樊李红黄进占昌友
Owner WUHAN UNIV OF TECH