Pyrenyl-containing radical initiator, and synthesis method and use thereof
A synthesis method and initiator technology, applied in chemical instruments and methods, preparation of organic compounds, organic chemistry, etc., can solve problems such as inapplicability of initiators
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Embodiment 1
[0042] Take a 150ml three-neck flask, mix 40ml of dichloromethane, 50.1mg (0.18mmol) of 4,4'-azo(4-cyanovaleric acid) (as shown in general formula B1), 92.9mg (0.40mmol) of pyrene Methanol (as shown in the general formula C1, where x=1), 8.6mg (0.07mmol) DMAP, 64.9mg (0.48mmol) HOBT were added to it successively, and a homogeneous solution was prepared under magnetic stirring. Then, under the conditions of ice-water bath and nitrogen protection, EDC.HCl / dichloromethane solution (86.3 mg (0.45 mmol) EDC.HCl dissolved in 10 ml of dichloromethane) was slowly added dropwise. After the dropwise addition was completed for 30 minutes, the ice-water bath was removed, and the temperature of the reaction system was raised to 30° C. for 24 hours of reaction. The reaction solution was filtered, and the filtrate was diluted to 100ml with dichloromethane. The solution was subjected to 3 times of 1M HCl (3×50ml), 3 times of saturated NaHCO 3 solution (3×50ml), three times of distilled wate...
Embodiment 2
[0045] The pyrene group-containing small molecule compound pyrenemethanol in Example 1 was replaced with pyrenebutanol (as shown by the general formula C1, where x=4), and the dosage was 104.3mg (0.38mmol); the dosage of dichloromethane was adjusted to 45ml, The amount of DMAP was adjusted to 19.5mg (0.16mmol), the amount of EDC.HCl was adjusted to 80.5mg (0.42mmol) without HOBT, the reaction temperature was adjusted to 25°C, and the reaction time was extended to 26 hours; other operating conditions were the same as in Example 1 . Obtain light yellow solid compound, productive rate is greater than 86%, and molecular structural formula is:
Embodiment 3
[0047] Take a 150ml three-neck flask, mix 70ml of dichloromethane, 50.3mg (0.18mmol) of 4,4'-azo (4-cyanovaleric acid), 97.1mg (0.42mmol) of pyrenemethylamine (as represented by the general formula C2) Shown, where x=1), 106.4mg (0.49mmol) Sulfo-NHS was added to it successively, and a homogeneous solution was prepared under magnetic stirring. Then, under the conditions of ice-water bath and nitrogen protection, EDC.HCl / dichloromethane solution (89.7mg (0.47mmol) EDC.HCl dissolved in 10ml of dichloromethane) was slowly added dropwise. After the dropwise addition was completed for 1 hour, the ice-water bath was removed, the temperature of the reaction system was raised to 35° C., and the reaction was carried out for 18 hours. The reaction solution was filtered, and the filtrate was diluted to 100ml with dichloromethane. The solution was subjected to 3 times of 1M HCl (3×50ml), 3 times of saturated NaHCO 3 solution (3×50ml), three times of distilled water (3×50ml), and the orga...
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