A kind of clean production method of 3‑(n, n‑disubstituted) aminoacetanilide compounds
A technology of aminoacetanilide and its production method, which is applied to the preparation of organic compounds, chemical instruments and methods, and the preparation of carboxylic acid amides. It can solve the problems of complex components, high content of organic poisons, and refractory degradation, and achieve the goal of reducing production costs. Effect
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Embodiment 1
[0038] Add 150 kg of m-acetamido aniline hydrochloride, 370 kg of water, and 85 kg of 17.7% ammonia water into the reaction kettle, stir well, and control the pH of the ammonia water to 6.5-7. Raise the temperature of the material to 90-95°C, add 200kg of 17.7% ammonia water, control the pressure of the reactor below 1.0MPa, pass 133kg of ethyl chloride and 165kg of 17.7% ammonia water from the reaction liquid, control the pH to 5-7, and the temperature to 95 Insulate and react at ~98°C for 18 hours, and use HPLC (high performance liquid chromatography) to measure the end point of sampling, and control the content of monoethyl (ie m-acetamido-N-ethylaniline) within 2%. After the reaction, add 400kg of water to dilute, adjust the pH to 7.0-7.5 with ammonia water, filter and wash with water when the temperature is cooled to below 40°C, and separate the N,N-diethyl-m-acetamidoaniline product (yield about 98% ) and mother liquor containing ammonium chloride.
[0039]
[0040] ...
Embodiment 2
[0042] Add m-acetaminoaniline hydrochloride 185kg, add water 451kg in the reaction kettle, throw 110kg17.7% ammonia water to control pH6.5~7, stir evenly, feed 165kg ethyl chloride and 210kg 17.7% ammonia water under the liquid surface, Raise the temperature to 85°C in about 1.5 hours, keep it warm for 1 hour, then raise the temperature to 95°C, control the pressure of the reactor below 1.0MPa, keep it at about 97°C for 20 hours, use HPLC (high performance liquid chromatography) to measure the end point of the sample, and control the single B base (i.e., m-acetamido-N-ethylaniline) content within 2%, control the monoethyl content within 2.5%, cool down to 70°C, continue stirring, let it cool down naturally, precipitate, after the material precipitates, stir for 2 hours Around 30°C, filter and wash with water to separate the N,N-diethyl-m-acetaniline product (yield about 96%) and the mother liquor containing ammonium chloride.
[0043] The separated ammonium chloride mother liquo...
Embodiment 3
[0045] Add 200kg of 2-amino-4-acetamidoanisole, 330kg of water, and 1.3kg of MF into the reaction kettle, stir well, raise the temperature of the materials to 80-85°C, and keep warm for 1 hour to dissolve. Add 188kg of 96% allyl chloride, add liquid ammonia to control the pH 5-6, and keep the temperature at 80-85°C for 6 hours. The HPLC method (high performance liquid chromatography) is used for sampling to measure the end point, and the control of monopropenyl (ie 3-N -allylamino-4-methoxyacetanilide) content within 4%. After the reaction, add 400kg of water to dilute, stir and crystallize for about 1 hour, until all crystallization is complete, cool down to below 50°C, filter, wash with water, and separate 3-(N,N-diallyl)amino-4-methoxy Acetanilide product (yield about 98%) and mother liquor containing ammonium chloride.
[0046] After the separated ammonium chloride mother liquor is physically filtered, it is passed into an adsorption oxidation reactor filled with DA201-...
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