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Preparation method of nano vesicles loaded with active substance of purple sweet potato skin

A technology of nanovesicles and active substances, applied in the field of preparation of nanovesicles, can solve the problems of easily ruptured vesicles, low drug loading rate, intermembrane fusion, etc., and achieve good biocompatibility and permeability, high loading The effect of drug rate, water solubility and targeting

Inactive Publication Date: 2016-07-06
仇颖莹
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0005] The technical problem mainly solved by the present invention: the amphiphilic block polymer can form a vesicle double-layer membrane, but the stability of the liposome-like vesicles currently used is poor, and it is easy to rupture and produce fusion between vesicle membranes , the problem of low drug loading rate when polymer vesicles are used as drug carriers, a method for preparing nanovesicles loaded with active substances from purple potato peels is provided. The present invention obtains active substances from purple potato peels, and then prepares amphiphilic Sexual block copolymers, using amphiphilic block copolymers, the purple potato active substances are loaded in the block copolymers to form nanovesicles, the nanovesicles prepared by the present invention have significant mechanical properties, and can be used as drug carriers Not only has a high drug loading rate, but also has good biocompatibility and permeability. The amphiphilic block copolymer loads the active substance of purple potato skin to prepare vesicles, which can greatly improve the water solubility of the active substance of purple potato skin. and targeting, and the application is more convenient and the effect is more significant

Method used

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Examples

Experimental program
Comparison scheme
Effect test

example 1

[0024] First, take 200g of purple potato skin, wash it, dry it, crush it, and sieve it to get 80 mesh purple potato skin powder, add 80% ethanol solution with a mass fraction of 10mL / g according to the liquid-to-material ratio, mix and extract at 350W power for 70s, and extract The solution was centrifuged at 2000r / min for 15min to remove the precipitate to obtain a supernatant, and the supernatant was centrifuged at 5000r / min for 15min to remove the precipitate to obtain a supernatant, and the supernatant was heated at 60°C Distill down for 40 minutes to obtain a concentrated solution; filter the concentrated solution with a 0.1 μm microfiltration membrane, collect the liquid after the microfiltration, filter the liquid after the microfiltration with a 0.05 μm ultrafiltration membrane, and collect the liquid after the filtrate, which is Active liquid of purple potato peel, for use; accurately weigh 8g ε-caprolactone, 8g polyethylene glycol, 50mL toluene and add it into a round...

example 2

[0027] First, take 250g of purple potato skin, wash it, dry it, crush it, and sieve it to obtain 90-mesh purple potato skin powder. Add 80% ethanol solution with a mass fraction of 11mL / g according to the liquid-to-solid ratio, mix and extract at 400W power for 80s, and extract The solution was centrifuged at 2500r / min for 18min to remove the precipitate to obtain a supernatant, and the supernatant was centrifuged at 6000r / min for 17min to remove the precipitate to obtain a supernatant, and the supernatant was heated at 65°C Distill down for 50 min to obtain a concentrated solution; filter the concentrated solution with a 0.2 μm microfiltration membrane, collect the liquid after the microfiltration, filter the liquid after the microfiltration with a 0.06 μm ultrafiltration membrane, and collect the liquid after the filtrate, which is Active liquid of purple potato skin, for use; accurately weigh 9g ε-caprolactone, 9g polyethylene glycol, 65mL toluene and add it into a round bot...

example 3

[0030] First, take 300g of purple potato skin, wash it, dry it, crush it, and sieve it to get 100 mesh purple potato skin powder, add 80% ethanol solution with a mass fraction of 12mL / g at a liquid-to-solid ratio, mix and extract for 90s under 450W power, and extract The solution was centrifuged at 3000r / min for 20min to remove the precipitate to obtain a supernatant, and the supernatant was centrifuged at 7000r / min for 20min to remove the precipitate to obtain a supernatant, and the supernatant was heated at 70°C Distill down for 60 minutes to obtain a concentrated solution; filter the concentrated solution with a 0.3 μm microfiltration membrane, collect the liquid after the microfiltration, filter the liquid after the microfiltration with a 0.08 μm ultrafiltration membrane, and collect the liquid after the filtrate, which is Active liquid of purple potato peel, for use; accurately weigh 10g ε-caprolactone, 10g polyethylene glycol, 80mL toluene and add it into a round bottom f...

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Abstract

The invention discloses a preparation method of nano vesicles loaded with an active substance of purple sweet potato skin, belonging to the field of vesicles. According to the preparation method, the active substance is acquired from the purple sweet potato skin, then amphipathic segmented copolymers are prepared, and the active substance of the purple sweet potato skin is loaded in the segmented copolymers to form the nano vesicles. The nano vesicles prepared by the preparation method have notable mechanical property, higher drug loading ratio as a drug carrier and good biological compatibility and penetrability, and the amphipathic segmented copolymers loaded with the active substance of the purple sweet potato skin are prepared into vesicles, which can improve the water solubility and targeting ability of the active substance of the purple sweet potato skin, are more convenient in application and have more remarkable effect.

Description

technical field [0001] The invention discloses a preparation method of nano-vesicles loaded with active substances of purple potato peel, belonging to the field of vesicles. Background technique [0002] As an important self-assembled nanostructure, vesicle is a kind of nano hollow sphere surrounded by a double membrane or multilayer membrane composed of some special molecules. In recent years, there are more and more applications in drug and gene delivery, nanoreactors, and surface modification of cell membranes. In principle, as long as amphiphilic molecules have both hydrophilic and hydrophobic parts, it is possible to aggregate into a vesicle structure. Therefore, many polymers with hydrophilic and hydrophobic properties can be used to prepare vesicle structures, such as block copolymers, which can be used to artificially synthesize vesicles. Compared with liposomal vesicles, polymer vesicles have many advantages, such as more stability, variable permeability, firm str...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): A61K9/127A61K47/34A61K36/39A61P1/14A61P35/00A61P39/06A61P1/16A61P9/12A61P9/10
CPCA61K9/1273A61K36/39A61K47/34
Inventor 仇颖莹王志慧
Owner 仇颖莹