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Spirulina polysaccharide eye drop, and preparation method and application thereof

A technology of spirulina polysaccharide and eye drops, which is applied in the direction of pharmaceutical formulations, medical preparations containing active ingredients, organic active ingredients, etc., to achieve the effect of simple preparation method, easy implementation, and broad application and development prospects

Inactive Publication Date: 2009-06-03
SHANDONG EYE INST
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

But at present, spirulina is only used in health products and food, so it is very necessary and important to develop spirulina and its bioactive substances for the treatment and prevention of ocular neovascularization

Method used

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Examples

Experimental program
Comparison scheme
Effect test

preparation example Construction

[0012] Step 1, preparation of spirulina polysaccharide: prepare the required spirulina polysaccharide of the present invention with the following process.

[0013] (1) Take the dry Spirulina platensis powder and add 95% ethanol, soak overnight; (2) Centrifuge and dry at 37°C, add double distilled water at a ratio of 1:12; (3) Adjust the pH to 10.0 with NaOH, and bathe in 80°C for 4 ~6h; (4) centrifuge, adjust pH to 7.0; (5) add 5% trichloroacetic acid for precipitation at 4°C overnight; (6) centrifuge, take supernatant, add 5% mass / volume Trichloroacetic acid precipitation for 3 hours; (7) Centrifuge, take the supernatant, add 5 times the volume of ethanol to precipitate, and overnight at 4°C; (8) Wash the precipitate twice with pure acetone, and vacuum freeze-dry; (9) Place the above precipitate in- Store at 20°C for more than 3 days to ensure the complete volatilization of acetone; (10) Add normal saline to fully dissolve the precipitate, centrifuge to remove undissolved sub...

Embodiment 1

[0018] First establish the animal model of alkali burn in C57 BL / 6 mice: the model animal is C57 BL / 66—8 weeks old, female mice, the mice are generally anesthetized, proparacaine hydrochloride eye drops are instilled in the eyes, and 3 μl 1N NaOH is directly dripped into the eyes. The surface of the mouse cornea was burnt with alkali for 30 seconds, and immediately rinsed with more than 20ml of normal saline.

[0019] The mouse alkali burn animal model established above was divided into two groups, the control group and the treatment group, and eye drops were applied immediately after burns. Each eye was given 5 μl of eye drops each time, 4 times a day, and the eye drops were treated for 7 days. The specific groups are as follows:

[0020] Control group: treated with Tiruo Compound Sodium Chloride Eye Drops.

[0021] Treatment group: Spirulina polysaccharide eye drops were used for eye drops.

[0022] After 7 days of treatment, the therapeutic effect was observed and compare...

Embodiment 2

[0024] When the polysaccharide concentration of the spirulina polysaccharide eye drops was 100 μg / ml, after 7 days, the corneal lesions of the mice were observed. It was found that the blood vessels in the control group mice grew significantly after alkali burns, and the growth area of ​​new blood vessels accounted for 1 / 2 to 3 of the entire cornea. / 4, while the 10μg / ml spirulina polysaccharide eye drops treatment group only had a small amount of new blood vessels growing near the limbus, accounting for about 1 / 15 of the entire corneal area. The paraffin-embedded section of the whole eyeball was taken and stained with HE. It can be seen that the corneal stroma of the mice in the control group had obvious edema after 7 days of alkali burn, and a large number of inflammatory cells infiltrated. Adhesion: In the treatment group, no obvious edema was found in the corneal stroma of the mice after 7 days of alkali burn, only individual inflammatory cell infiltration was seen, and no ...

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Abstract

The invention relates to an eye drop for preventing and treating angiogenesis diseases in the eye, particularly a spirulina polysaccharide eye drop, and a preparation method and an application thereof. The spirulina polysaccharide eye drop is prepared from spirulina polysaccharides extracted from spirulina powder. The eye drop comprises spirulina polysaccharides and artificial tears, wherein the concentration of spirulina polysaccharides is 100-500 mug / mL. The artificial tears can be replaced by Compound Sodium Chloride Eye drops. The invention prepares spirulina polysaccharides into an eye drop for treating and preventing angiogenesis diseases in the eye for the first time, and the preventing and treating effect is remarkably. The eye drop has the advantages of simple preparation method, convenient implementation, good therapeutic effect, and good application and development prospect.

Description

technical field [0001] The invention relates to an eye drop for preventing and treating eye neovascularization diseases, in particular to a spirulina polysaccharide eye drop and a preparation method and application thereof. Background technique [0002] Ocular neovascular disease has become the leading cause of blindness in my country, but its pathogenesis has not been fully understood, and there is a lack of effective treatment methods in clinical practice. The commonly used clinical methods for treating neovascularization are laser photocoagulation and photocoagulation combined with photodynamic methods, but their long-term efficacy is not good and the cost is high. More importantly, once neovascularization is formed, the damage and destruction to the eye will be irreversible. cause blindness in most patients. It is very necessary to find safe and effective bioactive substances with anti-neovascular activity for the prevention and treatment of eye neovascularization-relat...

Claims

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Application Information

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IPC IPC(8): A61K9/08A61K31/715A61P27/02
Inventor 杨玲玲谢立信王瑶周庆军刘廷
Owner SHANDONG EYE INST