Method for preparing aromatic diamine containing adamantane structure
A technology of aromatic diamine and adamantane, which is applied in the field of synthesis of adamantane derivatives, can solve the problems of high cost and low yield, and achieve the effect of low cost, high yield and stable process
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[0025] In one embodiment, the present invention provides a method for preparing an aromatic diamine containing an adamantane structure, the method may include the following steps:
[0026] (1) Under the protection of an inert gas and the presence of a catalyst, react a dihaloadamantane with an anilide to obtain an adamantane containing a diacylaminophenyl group; and
[0027] (2) Hydrolyzing the diacylaminophenyl-containing adamantane to obtain an aromatic diamine containing an adamantane structure.
Embodiment 1
[0029] This example involves the synthesis of 1,3-bis(4-aniline)adamantane using 1,3-dibromoadamantane and acetanilide as main raw materials.
[0030] The synthetic route of this embodiment is as figure 1 shown. Specifically, the synthesis method of this embodiment mainly includes the following two steps.
[0031] 1. Under nitrogen protection, add 440g of 1,3-dibromoadamantane into a 10L four-neck flask, then add 2.0L of dichloroethane, stir well, add 500g of acetanilide and stir well. Slowly add zinc dichloride and stir evenly, then heat up to reflux (internal temperature 80-85°C), first use a water separator to divide part of the water, and then use a reflux device. Reflux at this temperature for 24 hours. At this time, the lower layer is viscous solid, and the upper layer is dichloroethane solvent. Cool to room temperature, pour out the upper solvent, add 1.0LDMF (N,N-dimethylformamide) to raise the temperature to make the solid a fluid slurry, slowly pour the slurry int...
Embodiment 2
[0035] This example involves the synthesis of 1,3-bis(4-aniline)adamantane using 1,3-dichloroadamantane and acetanilide as main raw materials.
[0036] The synthesis method of this embodiment mainly includes the following two steps.
[0037] 1. Under nitrogen protection, add 420g of 1,3-dichloroadamantane into a 10L four-necked flask, then add 2.0L of dichloroethane, stir well, add 500g of acetanilide and stir well. Slowly add aluminum trichloride and stir evenly, then raise the temperature to reflux (internal temperature 80-85°C), first use a water separator to separate part of the water, and then use a reflux device. Reflux at this temperature for 24 hours. At this time, the lower layer is viscous solid, and the upper layer is dichloroethane solvent. Cool to room temperature, pour out the upper solvent, add 1.0LDMF to raise the temperature to make the solid a mobile slurry, slowly pour the slurry into 4.0L of stirred water, filter after stirring for 30 minutes, and obtain a...
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