Unlock instant, AI-driven research and patent intelligence for your innovation.

Preparation method of DL-panthenol

A technology of panthenol and crystal seed is applied in the field of preparation of DL-panthenol, which can solve the problem of high yield of DL-panthenol, and achieve the effects of being beneficial to industrial production, reducing precipitation and reducing energy consumption.

Pending Publication Date: 2022-04-08
安徽泰格生物科技有限公司
View PDF3 Cites 0 Cited by
  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

Disclosed a kind of crystallization method of DL-panthenol as CN110835309A, adopt DL-pantoate lactone and 3-amino propanol, under 65-85 ℃ condition, react synthetic DL-panthenol in dehydrated alcohol, then By optimizing the crystallization conditions, high-purity DL-panthenol solid products were prepared, but the highest yield of DL-panthenol was only 77%.

Method used

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
View more

Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0029] The present embodiment provides a kind of preparation method of DL-panthenol, comprises the following steps:

[0030] (1) Add ethyl acetate 820kg, DL-pantolactone 520kg (quality after converted purity) and 3-aminopropanol 300kg (quality after converted purity) successively in a dry and clean 5000L reactor, and heat up to 45°C, stirred and reacted for 6 hours to obtain DL-panthenol solution;

[0031] (2) Cool down the DL-panthenol solution to 20°C, add 100g of DL-panthenol, then continue to cool down to -5°C, after crystals appear, keep warm for 6h under stirring conditions for crystallization, and centrifuge to obtain DL-panthenol The wet product obtained 791kg of DL-panthenol solid after vacuum drying.

[0032] After testing, the specific rotation of the DL-panthenol product is 0, the residual content of 3-aminopropanol is ≤0.1%, the melting point is 65°C, the weight loss on drying is ≤0.5%, and the heavy metal content is ≤10ppm. DL- The panthenol content is 99.5%, a...

Embodiment 2

[0034] The present embodiment provides a kind of preparation method of DL-panthenol, comprises the following steps:

[0035] (1) Add ethyl acetate 845kg, DL-pantolactone 545kg (quality after converted purity) and 3-aminopropanol 300kg (quality after converted purity) successively in a dry and clean 5000L reactor, and heat up to 50°C, stirred and reacted for 4 hours to obtain DL-panthenol solution;

[0036] (2) Cool down the DL-panthenol solution to 10°C, add 100g of DL-panthenol, then continue to cool down to 5°C, after crystals appear, keep warm for 8h under stirring conditions for crystallization, and centrifuge to obtain DL-panthenol wet product, and obtained DL-panthenol solid 791kg after vacuum drying.

[0037] After testing, the specific rotation of the DL-panthenol product is 0, the residual content of 3-aminopropanol is ≤0.1%, the melting point is 65°C, the weight loss on drying is ≤0.5%, and the heavy metal content is ≤10ppm. DL- The panthenol content is 99.3%, and ...

Embodiment 3

[0039] The present embodiment provides a kind of preparation method of DL-panthenol, comprises the following steps:

[0040] (1) Add ethyl acetate 835.6kg, DL-pantolactone 535.6kg (mass after converted purity) and 3-aminopropanol 300kg (mass after converted purity) successively in a dry and clean 5000L reactor, The temperature was raised to 40°C, and the reaction was stirred for 5 hours to obtain a DL-panthenol solution;

[0041] (2) Cool down the DL-panthenol solution to 15°C, add 100g of DL-panthenol, and then continue to cool down to 0°C. After crystals appear, keep it warm for 7h under stirring conditions for crystallization, and centrifuge to obtain DL-panthenol wet product, and obtained DL-panthenol solid 796kg after vacuum drying.

[0042] After testing, the specific rotation of the DL-panthenol product is 0, the residual content of 3-aminopropanol is ≤0.1%, the melting point is 65°C, the weight loss on drying is ≤0.5%, and the heavy metal content is ≤10ppm. DL- The p...

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
Login to View More

PUM

No PUM Login to View More

Abstract

The invention provides a preparation method of DL-panthenol, which comprises the following steps: taking DL-pantoic acid lactone and 3-aminopropanol as raw materials, and carrying out acylation reaction in ethyl acetate or methyl isobutyl ketone to obtain a DL-panthenol solution; and carrying out cooling crystallization, solid-liquid separation and drying on the DL-panthenol solution to obtain a DL-panthenol solid. According to the method provided by the invention, the reaction can be carried out at a relatively low temperature, and the obtained DL-panthenol has relatively high purity and yield.

Description

technical field [0001] The invention belongs to the technical field of chemical production, and in particular relates to a preparation method of DL-panthenol. Background technique [0002] DL-panthenol is the precursor of vitamin B5, it is a kind of off-white powdery solid with a slight special smell and easy to absorb moisture. DL-panthenol is easily soluble in water, ethanol, methanol and propylene glycol, soluble in chloroform and ether, slightly soluble in glycerin, insoluble in vegetable oil, mineral oil and fat. Relatively stable in air and light. [0003] DL-Panthenol, D-Panthenol and D-Panthenol Ethyl Ether are widely used in cosmetics series, among which D-Panthenol and D-Panthenol Ethyl Ether are in liquid state, while DL-Panthenol can exist in solid form, so it is more convenient to use and transport Convenient and widely concerned. DL-Panthenol is a racemic mixture of L-Panthenol and D-Panthenol, which can be widely used in medicine, food and cosmetic industri...

Claims

the structure of the environmentally friendly knitted fabric provided by the present invention; figure 2 Flow chart of the yarn wrapping machine for environmentally friendly knitted fabrics and storage devices; image 3 Is the parameter map of the yarn covering machine
Login to View More

Application Information

Patent Timeline
no application Login to View More
Patent Type & Authority Applications(China)
IPC IPC(8): C07C231/02C07C231/24C07C235/08
Inventor 段小瑞周多翔刘升升方岩汪洪湖王新华
Owner 安徽泰格生物科技有限公司