Concentrated, water-soluble, granular plant growth regulator formulation and methods for use of same

Abstract

A water-soluble granular composition including at least 40% of at least one plant growth regulator, at least one binder, at least one disaccharide and at least one surfactant; as well as methods for making and using the composition are disclosed. The water-soluble granular composition advantageously improves preparation of a solid plant growth regulator formulation for spray application, as such composition swiftly dissolves, is easily metered for application, can be more highly concentrated and is dust-free. A presently preferred water-soluble granular composition includes at least 40% of at least one gibberellin as the plant growth regulator.

Description

FIELD OF THE INVENTION [0001] The present invention is directed to a water-soluble granular composition including at least 40% of at least one plant growth regulator, at least one binder, at least one disaccharide and at least one surfactant; as well as methods for making and using the composition. The water-soluble granular composition advantageously improves preparation of a solid plant growth regulator formulation for spray application, as such composition swiftly dissolves, is easily metered, can be more highly concentrated and is dust-free. A presently preferred water-soluble granular composition includes at least 40% of at least one gibberellin as the plant growth regulator. BACKGROUND OF THE INVENTION [0002] Plant growth regulators are useful for influencing a range of plant developmental processes including stem elongation, germination, dormancy, flowering, sex expression, enzyme induction, fruit size and quality, as well as leaf and fruit senescence. Plant growth regulators...

AI Technical Summary

Benefits of technology

[0015] The present invention is directed to a water-soluble granular composition including at least 40% of at least one plant growth regulator, at least one binder, at least one disaccharide and at least one surfactant; as well as methods for making and using the composition. The water-soluble granular composition advantageously improves preparation of a solid plant growth regulator formulation for spray application, as such composition swiftly dissolves, is easily metered, can be more highly concentrated and is dust-free for handling. A presently preferred water-soluble granular composition includes at least one gibberellin, polyvinylpyrrolidone, at least one disaccharide and at least one surfactant.

[0029] The invention is also directed to a method of enhancing the utilization of a solid plant growth regulator formulation for spray application comprising the step of formulating said plant growth regulator in a water-soluble granular formulation containing at least 40% of plant growth regulator. In the method, preparation of the formulation for spray application can be enhanced, since dust from the solid formulation can be eliminated upon transfer; accurate metering and rapid dissolution of the solid formulation can be attained. The method is also advantageous because the solid formulation contains twice the concentration of plant growth regulators as conventional formulations of plant growth regulators. A presently preferred formulation for use in the method is a water-soluble granular formulation which contains at least one plant growth regulator, at least one binder, at least one disaccharide and at least one surfactant. A presently most preferred formulation is a water-soluble granular formulation which contains at least one gibberellin, polyvinylpyrrolidone, lactose monohydrate and polyoxyethylene 20 monolaurate.

Problems solved by technology

Each of the conventional types of formulations has disadvantages, so research to provide improved plant growth regulator formulations continues.

Gibberellin solution formulations are disadvantageous in several respects.

The solutions, such as those of GA4+7 in propylene glycol, are less concentrated due to low solubility of actives, and have limited stability.

Of the currently used solvents, isopropyl alcohol and methyl alcohol offer severe disadvantages such as flammability and toxicity, which lead to restrictions in manufacturing, packaging, labeling, transportation, and warehousing of such solutions.

THFA, used in some of the formulations, is considered corrosive to the eye and skin.

Moreover, low solubility of gibberellins in propylene glycol does not permit preparation of high potency solution formulations.

These low strength solution formulations also require larger packaging, more storage space, and higher associated transportation, warehousing, and container disposal costs.

Due to very low solubility and undesirable hydrolysis, it has not been possible to formulate gibberellins in aqueous systems.

The primary disadvantage of wettable powder and soluble powder formulations is that they tend to produce dust upon handling, such as when pouring, transferring or measuring them.

This dust may pose health hazards.

Further, powder formulations tend to wet poorly and also solubilize slowly upon addition to water.

Formation of lumps or partially solubilized spray solutions will lead to uneven distribution of the plant growth regulator in the tank-mix with potential for reduced field performance.

Sometimes, foam in the spray tank caused by spray tank adjuvants can also affect wetting and solubility of wettable and soluble powders.

Wettable powder formulations will also leave undesirable insoluble residues both in the tank and on the sprayed foliage and fruit.

However, tablets deliver only between 0.1-1 gram of active ingredient per tablet.

They are not ideal for large-scale field operations.

Moreover, effervescent tablets are highly susceptible to humidity; may be slow to dissolve and are expensive.

The quality of water-dispersible granules is highly process- and active-ingredient-dependent; and can result in low yield recoveries, poor attrition resistance leading to dust potential, high manufacturing cost and poor dispersion.

Generally, sprays of dissolved water-dispersible granular formulations leave undesirable insoluble residues on the treated foliage and fruit.

Otherwise, product efficacy will be severely affected.

When water-dispersible granules are used, the grower often may not be able to realize if he had achieved the total solubility of the active ingredient in the spray solutions.

In addition, water-dispersible granules can become hardened over time and thus result in poor dispersibility and solubility of the active ingredient.

Dust and caking may be problems with certain water-dispersible granules and powder formulations.