Cyclopentadiene-N-(2-methylquinoline) titanium benzoic amide coordination compound as well as preparation method and application thereof
A cyclopentadienyl, benzamide titanium technology, applied in chemical instruments and methods, organic chemistry, metallocene and other directions, can solve the problems of difficult structural modification, poor stability, and limiting the practical application of metallocene catalysts
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[0051] Concrete preparation process is as follows:
[0052] 1. The general method of ligand synthesis
[0053] React 2-methyl-8-aminoquinoline with 1 equivalent of 4-substituted benzoic acid, and use 1 / 3 equivalent of triphenyl phosphite as a dehydrating agent, use xylene as a solvent, reflux for 6 hours, and concentrate , basic alumina or silica gel column chromatography, rinse with petroleum ether / ethyl acetate (5:1-10:1), the second effluent component is the product, and the solvent is removed to obtain a white solid N-(2-methyl quinoline) benzoic acid amide.
[0054] Second, the general method of synthesis of titanium complexes
[0055] At room temperature, the tetrahydrofuran solution of N-(2-methylquinoline)-benzoic acid amide was added dropwise to 1 equivalent of KH, and the reaction was stirred for 12 hours to obtain a yellow suspension. At -78°C, 1 equivalent of tetrahydrofuran solution of cyclopentadienyl titanium complex was added dropwise to the above suspension...
Embodiment 1
[0060] Example 1, Preparation of 4-methoxy-N-(2-methylquinoline) benzoic acid amide [ligand 1]
[0061]In 250ml flask, add 2-methyl-8-aminoquinoline (6.32g, 40mmol), 4-methoxybenzoic acid (6.08g, 40mmol) and dehydrating agent triphenyl phosphite (12.4g, 40mmol), Reflux in 100ml of xylene for 6 hours, remove the solvent in vacuo, and dissolve the residue with dichloromethane, perform basic alumina column chromatography, rinse with petroleum ether / ethyl acetate (10:1, v / v), The separated product was analyzed by thin layer chromatography, and the second eluent fraction (Rf=0.4) was collected, and the solvent was removed to obtain a white solid 4-methoxy-N-(2-methylquinoline) benzoic acid amide [ligand 1] 10.7 g, yield 92.0%. Melting point: 130-131°C.
[0062] The structural confirmation data are as follows:
[0063] 1 H NMR (CDCl 3 , 300MHz): δ10.77(s, N-H, 1H), 8.90(dd, J=7.5Hz, J=7.2Hz, 1H), 8.08(d, J=8.8Hz, 2H), 8.06(m, 1H) , 7.51(m, 2H), 7.36(d, J=8.5Hz, 1H), 7.06(d, J=...
Embodiment 2
[0067] Example 2, preparation of 4-methyl-N-(2-methylquinoline) benzoic acid amide [ligand 2]
[0068] Experimental procedure is with embodiment 1,2-methyl-8-aminoquinoline and 4-methylbenzoic acid condensation obtains white solid 4-methyl-N-(2-methylquinoline)-benzoic acid amide [ligand 2], rinsed with petroleum ether / ethyl acetate (10:1, v / v), separated the product by thin-layer chromatography, and collected the second elution fraction (Rf=0.4), with a yield of 91.2%. Melting point: 104-105°C.
[0069] The structural confirmation data are as follows:
[0070] 1 H NMR (CDCl 3 , 300MHz): δ10.84(s, N-H, 1H), 8.89(dd, J=7.0Hz, J=6.8Hz, 1H), 8.06(d, J=8.4Hz, 1H), 7.98(d, J= 8.8Hz, 2H), 7.54-7.47(m, 2H), 7.37-7.33(m, 1H), 7.22(d, J=8.4Hz, 2H), 2.78(s, CH 3 , 3H), 2.46(s, CH 3 , 3H).
[0071] 13 C NMR (CDCl 3 , 75MHz): δ162.0, 159.7, 154.3, 134.3, 133.1, 126.8, 126.0, 124.5, 122.4, 119.7, 118.3, 114.2, 112.9, 111.2, 22.4, 20.1.FT-IR (KBr, cm -1 ): 3345(m), 3050(w), 2913(w...
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