A preparation method for obtaining methane functionalized products based on combined iron/photocatalysis
A technology of functionalization and products, applied in the preparation of organic compounds, chemical instruments and methods, preparation of carboxylic acid nitrile, etc., can solve the problems of low methane carbon utilization efficiency, put the process into practice, slow progress, etc. A wide range of substrates, the effect of strong applicability
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Embodiment 1
[0024]
[0025] In the high pressure photoreactor, add magneton, benzylidene malononitrile (3.1mg, 0.02mmol), FeCl 3 ·6H 2 O (0.6 mg, 10% mol) and 1 mL of acetonitrile (CH 3 EN). Assemble the high pressure photoreactor, replace the gas atmosphere in the reactor with methane gas (5000kPa), operate 5 times, and then fill the reactor with methane gas to 5000kPa. Finally, irradiate with a 70W 365nm light source and stir at room temperature. After 14 hours, the reaction was diluted with ether, washed with deionized water, and the organic layer was concentrated in vacuo. The crude reaction product was purified and isolated by silica gel column chromatography to obtain the target product (colorless oil 3.2 mg, 95%). 1 H NMR (400MHz, CDCl 3 )δ7.48-7.32(m, 5H), 3.88(d, J=6.2Hz, 1H), 3.48(quint, J=6.9Hz, 1H), 1.68(d, J=7.1Hz, 3H); 13 C NMR (101MHz, CDCl 3 )δ138.20, 129.28, 128.88, 127.25, 111.98, 111.70, 41.22, 31.24, 17.79; HRMS (ESI - ):calcd for C 11 H 9 N 2 [M-H] - 16...
Embodiment 2
[0027]
[0028] In a high pressure photoreactor, add magnon, 2-(4-trifluoromethyl-benzylidene)malononitrile (4.4mg, 0.02mmol), FeCl3·6H2O (0.6mg, 10%mol) and 1mL acetonitrile (CH 3 EN). Assemble the high pressure photoreactor, replace the gas atmosphere in the reactor with methane gas (5000kPa), operate 5 times, and then fill the reactor with methane gas to 5000kPa. Finally, irradiate with a 70W 365nm light source and stir at room temperature. After 10 hours, the reaction was diluted with ether, washed with deionized water, and the organic layer was concentrated in vacuo. The crude reaction product was purified and isolated by silica gel column chromatography to obtain the target product (colorless oil 4.6 mg, 97%). 1 H NMR (400MHz, CDCl 3 )δ7.71(d,J=8.2Hz,2H),7.51(d,J=8.1Hz,2H),3.92(d,J=6.1Hz,1H),3.56(p,J=6.9Hz,1H) ,1.70(d,J=7.1Hz,3H). 13 C NMR (101MHz, CDCl 3 )δ141.96,131.21(q,J=33.3Hz),127.88,126.29(q,J=3.7Hz),123.76(q,J=275.7Hz),111.54,111.36,40.90,30.86,17.74.HR...
Embodiment 3
[0030]
[0031] In the high pressure photoreactor, add magneton, 2,2-dicyanovinyl-benzoic acid methyl ester (4.2mg, 0.02mmol), FeCl 3 ·6H 2O (0.6 mg, 10% mol) and 1 mL of acetonitrile (CH 3 EN). Assemble the high pressure photoreactor, replace the gas atmosphere in the reactor with methane gas (5000kPa), operate 5 times, and then fill the reactor with methane gas to 5000kPa. Finally, irradiate with a 70W 365nm light source and stir at room temperature. After 10 hours, the reaction was diluted with ether, washed with deionized water, and the organic layer was concentrated in vacuo. The crude reaction product was purified and isolated by silica gel column chromatography to obtain the target product (colorless oil 4.4 mg, 97%). 1 H NMR (400MHz, CDCl 3 )δ8.10(d,J=8.4Hz,2H),7.44(d,J=8.3Hz,2H),3.97-3.91(m,4H),3.54(p,J=6.9Hz,1H),1.69( d, J=7.1Hz, 3H). 13 C NMR (101MHz, CDCl 3 )δ166.39,142.98,130.76,130.52,127.44,111.66,111.43,52.34,41.06,30.84,17.74.HRMS(ESI - ):calcd for...
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