Organic radical modified DNA-cationic lipid complex and preparation method and application thereof
A cationic lipid and free radical technology, applied in electrical components, battery electrodes, circuits, etc., can solve the problems of difficult preparation of PTMA, reduce the molecular weight of polymers, reduce the performance of polymer organic free radical batteries, etc., and achieve a simple and feasible preparation process. , High physical and chemical stability, the effect of battery capacity is not easy to decay
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Embodiment 1
[0045] (1) Preparation of cationic lipids containing organic free radicals: Add 11-bromo-12 acid (1.33g, 5.0mmol) to a mixture containing EDC.HCl (1.0g, 5.2mmol) and DMAP (60mg, 0.50mmol) in an ice-water bath ) in dichloromethane (45mL), reacted with 4-hydroxy-TEMPO (1.20g, 5.7mmol) at room temperature for 12h, then washed three times with 50mL water, and the organic phase was washed with MgSO 4 The dried, rotary evaporated crude product was purified by a silica gel column to obtain 1.96 g of an orange solid (85%). The orange solid was subjected to reflux reaction in pyridine solvent for 48h, the pyridine was removed by rotary evaporation, and the cationic lipid containing free radical was obtained by precipitation in diethyl ether [attached figure 2 Lipid(1)];
[0046] (2) Preparation of DNA-cationic lipid complexes modified by organic radicals (attached image 3 shown): Dissolve 2.0mmol of free radical-containing cationic lipid in 5ml THF, slowly add to deionized water to...
Embodiment 2
[0051] (1) Preparation of cationic lipids containing organic free radicals: Add 11-bromo-12 alcohol (1.33g, 5.0mmol) to a mixture containing EDC.HCl (1.0g, 5.2mmol) and DMAP (60mg, 0.50mmol) in an ice-water bath ) in dichloromethane (45mL), reacted with 3-carboxy PROXYL (1.20g, 5.7mmol) at room temperature for 12h, then washed three times with 50mL of water, and the organic phase was washed with MgSO 4 Drying. The crude product obtained by rotary evaporation was purified by a silica gel column to obtain 1.96 g of an orange solid (85%). The above product was reacted with pyridine for 48 hours under reflux, the pyridine was removed by rotary evaporation, and the cationic lipid containing free radicals was obtained by precipitation in diethyl ether [attached figure 2 lipid(L1-P)] in
[0052] (2) Preparation of DNA-cationic lipid complexes modified by organic radicals (attached image 3): Dissolve a small amount of free radical-containing cationic lipid [lipid(L1-P)] in 10ml TH...
Embodiment 3
[0057] (1) Preparation of cationic lipids containing organic free radicals: react 11-bromo-12 acid with L-glutamic acid-α,γ-dimethyl ester hydrochloride [Glu(OMe)-OMe·HCl], and the product desorbs Remove methyl to obtain carboxyl-containing product, react with 4 hydroxyl TEMPO then, prepare the lipid containing 2 TEMPO free radicals in each lipid molecular structure according to the method in example 1 (attachment figure 2 Lipid(L2-T) in.
[0058] (2) Preparation of DNA-cationic lipid complexes modified by organic radicals (attached image 3 ): Dissolve a small amount of free radical-containing cationic lipid [Lipid(L2-T)] in 10ml THF (30wt%), slowly add to deionized water to form a uniform and transparent aqueous solution (5wt%); 0.5gDNA-Na (base pair 10000) was dissolved in 100mL water (0.5wt%), and then the DNA-Na solution was slowly added to the lipid aqueous solution, the molar ratio of phosphate to lipid was 1.5, stirred for 24h, and the DNA-cation was precipitated Th...
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