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Method for preparing radix astragali temperature-sensitive gel for treating helicobacter pylori positive gastric ulcers

A technology of Helicobacter pylori and temperature-sensitive gel, which is applied in the directions of non-active ingredient medical preparations, active ingredients-containing medical preparations, pharmaceutical formulas, etc. Treatment requirements and other issues to achieve the effect of prolonging the stagnation time, maintaining drug concentration, and delaying drug release

Inactive Publication Date: 2016-08-17
陈建峰
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0005] The technical problem mainly solved by the present invention: for the current treatment of H. The bioavailability is low, and it may lead to the problem that the drug concentration at the lesion cannot meet the treatment requirements. A preparation method of Astragalus thermosensitive gel for Helicobacter pylori positive gastric ulcer is provided. The invention uses Astragalus as raw material, by adding The citrate buffer solution controls the pH to be 6-8, and lecithin is added to the astragalus solution to react to obtain astragalus ethanol plastid suspension, and chitosan, glycerin and poloxamer are added to the suspension to react at low temperature. Temperature-sensitive gel, adding potassium sorbate preservative to the temperature-sensitive gel can keep it for a long time. Astragalus temperature-sensitive gel is stored at low temperature and is liquid at low temperature. When it enters the human body, it forms a semi-solid gel state in the stomach , can be filled in the tissue gap, prolonging the stagnation time of the astragalus thermosensitive gel in the stomach, delaying drug release, and helping to maintain local drug concentration, suitable for local treatment

Method used

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Examples

Experimental program
Comparison scheme
Effect test

example 1

[0017] First weigh 5g of lecithin and add it to a 250mL beaker with 100mL of ethanol, stir for 3min to obtain an ethanol solution of lecithin; weigh 10g of astragalus and add it to a 500mL beaker, put the beaker into a water bath to keep the temperature at 36°C, and add Add 200mL of citrate buffer solution with a pH of 6 into the beaker, and add the lecithin ethanol solution dropwise at 5mL / min into the 500mL beaker while stirring, then put the beaker into an ice-water bath, control the temperature at 0°C, and react 2h, and then use 180w ultrasonic wave for 10min to obtain astragalus ethanolic plastid suspension; add 20g chitosan to the above astragalus ethanolic plastid suspension, control the temperature in the water bath at 65°C, stir for 10min, and then add 30mL Glycerin, 30mL poloxamer, controlled temperature at 65°C, stirred and reacted for 12h, cooled the reaction solution to room temperature naturally to obtain a gel; added 1g of potassium sorbate to the above gel, cont...

example 2

[0020] First weigh 8g of lecithin and add it to a 250mL beaker with 150mL of ethanol, stir for 4min to obtain an ethanol solution of lecithin; weigh 15g of astragalus and add it to a 500mL beaker, put the beaker into a water bath to keep the temperature at 38°C, and add Add 250mL of citrate buffer solution with a pH of 7 into the beaker, add the ethanol solution of lecithin mentioned above dropwise into the 500mL beaker at 6mL / min while stirring, then put the beaker into an ice-water bath, control the temperature at 3°C, and react 2.5h, then use 180w ultrasonic wave for 15min to obtain the astragalus ethanol plastid suspension; add 25g chitosan to the above astragalus ethanol plastid suspension, control the temperature in the water bath at 70°C, stir for 11min, and then add 40mL glycerin, 40mL poloxamer, control the temperature at 70°C, stir and react for 13h, naturally cool the reaction solution to room temperature, and obtain a gel; add 1.5g potassium sorbate to the above ...

example 3

[0023] First weigh 10g of lecithin and add it to a 250mL beaker with 200mL of ethanol, stir for 5min to obtain an ethanol solution of lecithin; weigh 20g of astragalus and add it to a 500mL beaker, put the beaker into a water bath to keep the temperature at 40°C, and add Add 300mL of citrate buffer solution with a pH of 8 into the beaker, and add the ethanol solution of lecithin mentioned above into the 500mL beaker dropwise at 8mL / min while stirring, control the temperature at 5°C in an ice-water bath, react for 3h, and then use a 200w ultrasonic wave to sonicate 20min, to obtain astragalus ethanol plastisome suspension; add 30g chitosan to the above suspension, control the temperature in a water bath at 75°C, stir for 12min, then add 50mL glycerin and 50mL poloxamer to it successively, control the temperature at Stir at 75°C for 14 hours, cool the reaction solution to room temperature naturally to obtain a gel; add 2 g of potassium sorbate to the above gel, control the temper...

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PUM

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Abstract

The invention discloses a method for preparing radix astragali temperature-sensitive gel for treating helicobacter pylori positive gastric ulcers, and belongs to the field of temperature-sensitive high polymer material gelatinizing agents. The radix astragali temperature-sensitive gel is prepared from radix astragali, a citrate buffer solution is added to control the pH to range from 6 to 8, lecithin is added into the radix astragali solution for reacting, radix astragali ethyl alcohol plastid suspension is obtained, chitosan, glycerinum and poloxamer are added into the suspension for low-temperature reacting, and temperature-sensitive gel can be obtained; a potassium sorbate corrosion remover is added into the temperature-sensitive gel, so that the radix astragali temperature-sensitive gel is preserved for a long time, the radix astragali temperature-sensitive gel is preserved at low temperature and is in a liquid state at low temperature, the radix astragali temperature-sensitive gel is in a semi-solid gel state in the stomach after entering the human body, tissue clearances can be filled with the radix astragali temperature-sensitive gel, the stagnation time of the radix astragali temperature-sensitive gel in the stomach is prolonged, medicine release can be delayed, the local medicine liquid concentration can be maintained, and the radix astragali temperature-sensitive gel is suitable for local treatment.

Description

technical field [0001] The invention discloses a preparation method of an astragalus temperature-sensitive gel for treating Helicobacter pylori-positive gastric ulcer, and belongs to the field of temperature-sensitive polymer material gels. Background technique [0002] Ulcer disease or peptic ulcer is a common digestive tract disease that can occur in the esophagus, stomach or duodenum, and can also occur near the gastric-cavity anastomosis or diverticulum containing gastric mucosa. The main causes are: Helicobacter pylori infection, drugs and dietary factors, clinical symptoms mainly include: epigastric pain is the main symptom of this disease. At present, the drugs for the treatment of hypertension mainly include drugs that reduce damage factors: such as antacids, anticholinergic drugs, proglumide, etc., and drugs that protect the gastric mucosa at the same time: such as sucralfate, bismuth, and ketone etc. and the application of antibiotics. The above drugs are all oral...

Claims

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Application Information

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IPC IPC(8): A61K9/06A61K36/481A61K47/36A61K47/10A61K47/24A61K47/34A61P1/04
CPCA61K9/06A61K36/481A61K47/10A61K47/24A61K47/36
Inventor 陈建峰孟浩影
Owner 陈建峰