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An enzyme-responsive magnetic nanoparticle and its preparation method and application

A magnetic nanoparticle, enzyme-responsive technology, applied in the field of medicine, to achieve the effect of strong targeting, rich sources and good use effect

Active Publication Date: 2018-05-15
ZHENGZHOU UNIV
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0004] Currently, the magnetic Fe 3 o 4 @Cu 2-x S is the magnetic targeting material and photosensitizer, gelatin and sodium alginate are the composite capsule materials, the construction of new enzyme-responsive magnetic nanoparticles, and its application in tumor targeting therapy have not yet been published.

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0014] In concrete implementation, the present invention is realized by the following steps:

[0015] 1) Synthesis of Fe 3 o 4 Nanoparticles: Weigh FeSO 4 ·7H 2 O 3.36g and FeCl 3 ·6H 2 O 3.2g, dissolved in 80mL ultrapure water, in N 2 Protect and stir at 80°C for 30 minutes, then add 8mL of ammonia water, the solution turns black, continue to stir for 30 minutes, weigh 1.6g of citric acid and dissolve it in 3.2mL of ultrapure water, then add to the above black solution, heat up to 95°C, React for 90 minutes, magnetically separate to obtain a precipitate, wash the precipitate 3 times, and vacuum dry at 60°C to obtain Fe 3 o 4 Nanoparticles;

[0016] 2) Synthesis of magnetic Fe 3 o 4 @Cu 2-x S nanomaterials: Weigh 3.6mmoL sublimated sulfur and dissolve it in 2.4mL oleylamine, add 0.16mmoL Fe 3 o 4 In 8 mL of cyclohexane containing nanoparticles, stir at 70°C for 10 min to form sublimated sulfur and Fe 3 o 4 cyclohexane mixed solution; in addition, 0.4mmoL copper ...

Embodiment 2

[0019] The present invention can also be realized by the following steps in concrete implementation:

[0020] 1) Synthesis of Fe 3 o 4 Nanoparticles: Weigh FeSO4 ·7H 2 O 4.2g and FeCl 3 ·6H 2 O 4.0g, dissolved in 100mL ultrapure water, in N 2 Protect and stir at 80°C for 30 minutes, then add 10mL of ammonia water, the solution turns black, continue to stir for 30 minutes, weigh 2g of citric acid and dissolve it in 4mL of ultrapure water, then add to the above black solution, heat up to 95°C, and react for 90min , magnetically separated to obtain a precipitate, which was washed three times with water, and dried under vacuum at 60°C to obtain Fe 3 o 4 Nanoparticles;

[0021] 2) Synthesis of magnetic Fe 3 o 4 @Cu 2-x S nanomaterials: Weigh 4mmoL sublimated sulfur and dissolve it in 3mL oleylamine, add 0.2mmoL Fe 3 o 4 In 10 mL of cyclohexane containing nanoparticles, stir at 70°C for 10 min to form sublimated sulfur and Fe 3 o 4 cyclohexane mixed solution; in additi...

Embodiment 3

[0024] In concrete implementation, the present invention is realized by the following steps:

[0025] 1) Synthesis of Fe 3 o 4 Nanoparticles: Weigh FeSO 4 ·7H 2 O 50.4g and FeCl 3 ·6H 2 O 4.8g, dissolved in 120mL ultrapure water, in N 2 Protect and stir at 80°C for 30 minutes, then add 10mL of ammonia water, the solution turns black, continue to stir for 30 minutes, weigh 2.4g of citric acid and dissolve it in 4.8mL of ultrapure water, then add to the above black solution, heat up to 95°C, React for 90 minutes, magnetically separate to obtain a precipitate, wash the precipitate 3 times, and vacuum dry at 60°C to obtain Fe 3 o 4 Nanoparticles;

[0026] 2) Synthesis of magnetic Fe 3 o 4 @Cu 2-x S nanomaterials: Weigh 4.8mmoL sublimated sulfur and dissolve it in 3.6mL oleylamine, add 0.24mmoL Fe 3 o 4 In 12 mL of cyclohexane containing nanoparticles, stir at 70°C for 10 min to form sublimated sulfur and Fe 3 o 4 cyclohexane mixed solution; in addition, 0.6mmoL copp...

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Abstract

The invention relates to an enzyme-responsive magnetic nanoparticle and its preparation method and application, which can effectively solve the problem of the preparation of the enzyme-responsive magnetic nanoparticle and its application in tumor treatment as a magnetic hyperthermia medium and a drug delivery carrier. The method is as a drug The carrier system uses Fe3O4@Cu2‑xS composite nanomaterials as magnetic targeting materials and photosensitizers, gelatin and sodium alginate as composite capsule materials, and the magnetic Fe3O4@Cu2‑xS composite nanomaterials are first prepared by chemical co-precipitation. Fe3O4 nanoparticles , and then load Cu2‑xS on the surface of Fe3O4 nanoparticles to obtain a core-shell Fe3O4@Cu2‑xS composite material. Finally, gelatin and sodium alginate are used as composite capsule materials, and the carrier and anticancer drugs are prepared by complex coacervation method Forming an enzyme-responsive magnetic nanoparticle, the raw material source of the present invention is abundant, the cost is low, the quality is good, the targeting property is strong, and the use effect is good, which is a great innovation in tumor treatment drugs.

Description

technical field [0001] The invention relates to medicine, in particular to an enzyme-responsive magnetic nanoparticle and its preparation method and application. Background technique [0002] Tumor is one of the most harmful diseases to humans in the world today. Due to its complex pathogenesis and large gene mutations, traditional therapeutic drugs have little effect in reducing the incidence and mortality of tumors. Near-infrared light-mediated photothermal therapy proposed in recent years can eliminate tumor tissue at a specific point and has low side effects on normal tissue, which provides a new way for tumor treatment. The latest reported semiconducting copper sulfide (Cu 2-x S) Nanoparticles, with simple preparation process, low cost, outstanding photothermal stability and good biocompatibility, have become a research hotspot in the field of nanomedicine. [0003] Tumor invasion and metastasis are the main biological characteristics of malignant tumors and have beco...

Claims

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Application Information

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Patent Type & Authority Patents(China)
IPC IPC(8): A61K41/00A61K9/51A61K47/42A61K47/36A61K31/704A61P35/00
Inventor 张振中祝侠丽黄河清张英杰侯琳张慧娟李鸿基
Owner ZHENGZHOU UNIV