The invention relates to a Chinese medicament for treating hyperprolactinemia and a preparation method thereof. The medicament is prepared from ten Chinese medicinal materials, namely radix bupleuri, white peony roots, angelica, nutgrass galingale rhizome, cortex moutan radicis, gardenia, roses, malt, herba ecliptae and glossy privet fruits. The medicament has the efficacy in soothing liver, relieving upset, nourishing Yin and blood, clearing heat and relieving restlessness, and is used for premenstrual tension syndrome, infertility accompanied by serum prolactin increase, as well as people with liver depression, heat transformation, deficiency of yin-fluid and blood. Symptoms include irregular menstruation, amenorrhea, no impregnation long after marriage, painful chest and hypochondrium or mammary swelling pain, light headedness, vexation, irascibility, agrypnia, dreaminess, mouth-throat dryness, waist-knee lassitude, red tongue with thin yellow fur or thin white dry fur and string-like rapid pulse. Clinical verification results show that the medicament is safe, effective and free from toxic or side effects on human bodies.