Fluorene carbazole derivative as well as preparation method and application thereof
A technology of fluorenocarbazole and derivatives, which is applied in the field of fluorenocarbazole derivatives and their preparation, can solve the problems of difficult synthesis and constraints, and achieve the expansion of conjugated structure, compact configuration, high thermal stability and electrogenicity. The effect of the characteristic
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Embodiment 1
[0048] Embodiment 1: the synthesis of intermediate fluorenocarbazole
[0049]
[0050] S1. In a 250mL three-necked flask, put 4-bromo-9,9-dimethyl-9H-fluorene (8.20g, 30mmol), 2-chloroaniline (4.59g, 36mmol), triphenylphosphine (0.04g , 0.15mmol), sodium tert-butoxide (8.65g, 90mmol), add 80mL ethanol and 40mL water, under nitrogen atmosphere, add tris(dibenzylideneacetone) dipalladium (0.27g, 0.3mmol), at 70°C Reaction 1-4h, liquid phase monitoring 4-bromo-9,9-dimethyl-9H-fluorene reaction is complete, add water to quench the reaction, separate liquid, concentrate the organic phase, rinse with petroleum ether through a silica gel column, rinse The solution was concentrated to obtain 9.02 g of N-(2-chlorophenyl)-9,9-dimethyl-9H-fluoren-4-amine as a colorless transparent oil, with a yield of 94% and a purity of 99.85%.
[0051] S2. In a 100mL three-necked flask, put the above-mentioned N-(2-chlorophenyl)-9,9-dimethyl-9H-fluorene-4-amine (5.67g, 20mmol), tri-tert-butylphosph...
Embodiment 2
[0052] Embodiment 2: the synthesis of compound (4)
[0053]
[0054] S3. In a 250mL three-necked flask, put the above-mentioned fluorenylcarbazole (4.25g, 15mmol), 5-bromo-2-iodopyridine (5.67g, 20mmol), 18-crown-6 (0.79g, 3mmol), Potassium carbonate (10.36g, 75mmol), add 75mL dimethylacetamide, under nitrogen atmosphere, add cuprous iodide (0.57g, 3mmol), react at 160°C for 4-8h, monitor the completion of the reaction in liquid phase, cool to room temperature, washed with water, filtered, and the filter cake was beaten again with 3-5 times of ethyl acetate, and then heated with a 10:1 ethyl acetate: ethanol mixed solvent to obtain white powdery intermediate 12-( 5-bromopyridin-2-yl)-fluorenocarbazole 5.47g, yield 83%.
[0055] S4. In a 100mL three-necked flask, put the above-mentioned intermediate 12-(5-bromopyridin-2-yl)-fluorenocarbazole (2.20g, 5mmol), 4,4-dimethyldiphenylamine (1.78g, 9mmol), tri-tert-butylphosphine tetrafluoroborate (0.06g, 0.2mmol), sodium tert-but...
Embodiment 3
[0057] Embodiment 3: the synthesis of compound (9)
[0058]
[0059] The 5-bromo-2-iodopyridine (5.67g, 20mmol) in Example 2 was replaced by 4-bromo-4'-iodo-1,1'-biphenyl (7.18g, 20mmol), 4,4-bis Methyldiphenylamine (1.78g, 9mmol) is replaced by diphenylamine (1.52g, 9mmol), and other synthetic processes are the same as in Example 2 (the intermediates of each corresponding step can be different, but other reactants, mol ratios, and reaction conditions are identical ) to obtain 2.50 g of compound (9) in the form of white powder, with a yield of 90%.
[0060] Mass spectrometer MALDI-TOF-MS (m / z) = 602.7803, theoretical molecular weight: 602.7810; Anal.Calcd forC 45 h 34 N 2 (%): C 89.67, H 5.69, N 4.65, Found: C 89.69, H 5.68, N 4.64.
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