The application provides an internal gold
peroxide complex, a preparation method and application thereof, and a structure formula of the internal gold
peroxide complex is as a compound of formula (I) or a pharmaceutically acceptable salt thereof: The compound of formula (I) has photo-reactivity, under light conditions, the
peroxide bond is cleaved, and a carbon free radical with
biological activity is converted subsequently, can be combined with biological macromolecular proteins,
DNA to destroy related biological functions, and plays an anticancer role; the compound can also contain a
small molecule drug residue, and the released
small molecule drug can enhance the
antitumor activity in vivo.