The application relates to an
aryl boron compound, a preparation method and application thereof, and a pharmaceutical composition, which is used for
tumor imaging, has high
fluorescence quantum efficiency through intramolecular charge transfer, and can be connected to different antibodies through Q3 under a certain concentration, and can accurately target corresponding tumors according to different antibodies. The
boron drug preparation can be used for
boron neutron capture therapy to kill
tumor cells. The compound has a better killing effect, and the compound is targeted to
tumor cells through
antigen-
antibody interaction. After the boron-10
drug is gathered at a
tumor site,
neutron radiation is generated, a
nuclear reaction is triggered to release alpha particles and 7 Li particles kill cells, and the ranges of the two particles are about 10 mu m. High-energy-density heavy ions break the double
helix structure of
DNA in
tumor cells, so that the cells cannot be repaired and die completely, and the distance of 10 mu m avoids damage to normal cells and tissues.