6 results about "Famoxadone" patented technology

The invention relates to novel acridine spiroisoxazole compounds, a preparation method thereof and application of the novel acridine spiroisoxazole compounds in antifungal drugs. The novel acridine spiroisoxazole compounds have the antibacterial activity of 36 compounds, and the 36 compounds have the inhibiting effect on botrytis cinerea, parasite scalaria, rhizoctonia solani, fusarium graminearum and candida albicans. The antifungal biological activity result shows that the compound series all show obvious antibacterial activity. The compound is determined as a broad-spectrum antibacterial candidate due to the comprehensive antibacterial characteristics of the compound, and the EC50 value (5.0 + / -0.4 mu g / mL) of H35 shows 1.5 times, 2.2 times and 3.2 times of titer advantages compared with positive control drugs famoxadone (7.6 mu g / mL), chlorothalonil (11.1 mu g / mL) and carbendazim (15.9 mu g / mL) respectively. The spiro structure of the compound can significantly improve the antibacterial activity of the compound, the preliminary mechanism research target shows that the compound is related to fungal membrane damage, and in addition, the compound H35 has protection and treatment effects on botrytis cinerea infection in corn, which shows that the compound H35 has agricultural application potential.

The invention relates to a novel acridinyl-containing tetrahydronaphthalene spiro isoxazoline compound, a preparation method thereof and application of the novel acridinyl-containing tetrahydronaphthalene spiro isoxazoline compound as an antifungal drug. The novel acridinyl-containing tetrahydronaphthalene spiroisoxazoline compound has an inhibition effect on parasite sphaerospora, botrytis cinerea, rhizoctonia solani, fusarium graminearum and candida albicans in the antifungal activity of the novel acridinyl-containing tetrahydronaphthalene spiroisoxazoline compound. An antifungal biological activity result shows that the compound shows remarkable antifungal activity, has comprehensive antifungal characteristics and is determined as a broad-spectrum antifungal candidate, the EC50 value of the compound to parasitic powdery spores is superior to that of a positive control drug chlorothalonil, and the compound shows about 12 times and 25 times of titer advantages compared with famoxadone and carbendazim respectively. The spiro structure and multiple active groups of the compound can significantly improve the antifungal activity of the compound, and in addition, the compound has protection and treatment effects on powdery parasitic spore infection in corn, which shows that the compound has agricultural application potential.

A composition including a compound of formula (I)and one or more mitochondrial electron transport system complex III inhibitor(s) selected from the group consisting of azoxystrobin, coumoxystrobin, enoxastrobin, flufenoxystrobin, picoxystrobin, pyraoxystrobin, pyraclostrobin, mandestrobin, pyrametostrobin, triclopyricarb, kresoxim-methyl, trifloxystrobin, dimoxystrobin, fenaminstrobin, metominostrobin, orysastrobin, famoxadone, fluoxastrobin, fenamidone, pyribencarb, metyltetraprole, cyazofamid, amisulbrom, fenpicoxamid, and florylpicoxamid.

The invention discloses a vacuum rake dryer for famoxadone bactericide production, and belongs to the field of dryers. The vacuum rake dryer for famoxadone bactericide production comprises a shell and a hollow rotating shaft rotationally connected to the interior of the shell, a first hollow shaft and a second hollow shaft are arranged in the rotating shaft, and a plurality of rake tooth assemblies are arranged on the rotating shaft; the rake tooth assembly comprises a rake tooth shaft fixedly arranged on the rotating shaft, a connecting shaft rotationally connected to the rake tooth shaft, rake teeth arranged at one end of the connecting shaft and a transmission assembly arranged at the other end of the connecting shaft, and the rake teeth are in sliding contact with the inner wall of the shell; and a driving assembly for controlling the rake tooth shaft to rotate is arranged in the second hollow shaft. By synchronously adjusting the inclination angles of all the rake teeth, the characteristics of materials and the requirements of all drying stages can be matched, and the drying rate and uniformity are optimized; and meanwhile, the rake tooth angle can be conveniently adjusted in real time according to the actual working condition of the dried materials, and the applicability of the dryer to various materials is improved.

The present application relates to a kind of fungicidal compositions containing famoxadone and carvacol, and the effective component is the binary complex of famoxadone and carvacol.The mass ratio of famoxadone and carvacol is 1-20:30-5, and the mass fraction ratio of effective component famoxadone and carvacol in preparation is 6%-50%.The dosage form of the fungicidal composition described in the present application is emulsifiable concentrate, suspension concentrate, water emulsion, microemulsion and water dispersible granule.The fungicidal composition is suitable for preventing and treating various powdery mildew, rust, leaf blight, net blotch, downy mildew, early and late blight of fruit trees, vegetables, ornamental plants, crops, etc., and has good protective and curative effects on early and late blight of tomato, etc.

A succinate sulfonate-containing fungicide, and a preparation method therefor and a use thereof. The fungicide at least comprises the following components: (a) at least one chemically active substance for controlling crop fungal diseases, the chemically active substance being selected from one or more of tebuconazole, trifloxystrobin, prothioconazole, cyazofamid, cymoxanil, famoxadone, difenoconazole, pyraclostrobin, boscalid, and fludioxonil; (b) at least one succinate sulfonate; and (c) an auxiliary agent, the auxiliary agent comprising at least one of a carrier, a disintegrant, a binder, a rheology modifier, a dispersant, a wetting agent, a defoaming agent, a thixotropic agent, an antifreeze agent, a preservative, a thickener, a solvent, and an emulsifier. By optimizing a fungicide formulation system, the utilization rate of fungicidal agricultural active substances is improved, thereby achieving the objective of reducing dosage while enhancing efficacy; and the fungicide has high market promotion value.