A whitening nanocomposition, a preparation method therefor, and use thereof. The whitening nanocomposition comprises an
active ingredient and a nanocarrier. The
active ingredient is coated and / or adsorbed by the nanocarrier. The
active ingredient comprises the following components: 1-15 parts by weight of α-
arbutin, 1-15 parts by weight of
nicotinamide, 1-10 parts by weight of 3-o-ethyl
ascorbic acid, 0.1-1 part by weight of a Centalla asiatica extract, and 1-5 parts by weight of
retinyl palmitate. The nanocarrier comprises the following components: 5-10 parts by weight of an emulsifier, 5-20 parts by weight of a
polyol, 0.1-5 parts by weight of a
phospholipid, and 40-60 parts by weight of water. The whitening nanocomposition has good
skin permeability and retention performance and enables high-concentration enrichment, prolonged retention, and sustained release or
controlled release within a
target tissue, so as to be effectively taken in by target cells, thereby improving
bioavailability and enhancing the whitening effect.