The invention discloses a benzofuran compound and a medical application thereof, and relates to a compound and an application thereof. A general formula of the compound is as shown in the specification, wherein R and R' are independently selected from hydrogen, methyl, ethyl or tertiary butyl; or the R and R', together with nitrogen atoms connected to the R and R', form pyrrolidyl, piperidyl or morpholinyl. The compound, disclosed by the invention, through an enzyme inhibiting property efficacy and other biochemical parameters thereof, can achieve an effective treatment effect by an expected usable dosage range which is about 0.01-10mg / kg per day; the compound is bound or embedded in a soluble and / or biodegradable polymer and is coated on a Stent's impression material; such polymer contains polyvinylpyrrolidone, polyhydroxy-propyl isobutylene amide-phenol, and a cross-linked or amphiphilic block copolymer of hydrogel.