The invention relates to a heterocyclic asymmetric aromatic dithioether compound and application thereof in herbicide preparation. As shown as in the formula (I), the compound has inhabitation effect to arabidopsis thaliana acetolactate synthase (AHAS) in vitro, has inhabitation effect to rape root length in vivo, has weeding effect for rape and redroot amaranth in potted plant tests, and can be used for preparing novel herbicides containing targeted AHAS. In the formula (I), when X represents S, R1 represents H, C1-C3 alkyl, C1-C3 acylamino, phenyl, hydroxylphenyl phenyl and ortho-C1-C3 alkoxy phenyl, R2 represents H, ortho-nitryl or para-nitryl, ortho-halogen or para-halogen, ortho-C1-C3 alkyl or para-C1-C3 alkyl, ortho-C1-C3 carbalkoxy, para-C1-C3 alkoxy and 3,4-benzo; and when X represents O, R1 represents H, phenyl, hydroxylphenyl phenyl, ortho-C1-C3 alkoxy phenyl, 4-pyridyl and 3-pyridyl, and R2 represents H, ortho-nitryl, para-C1-C3 alkyl and ortho-C1-C3 carbalkoxy.