The present application provides a
carvacrol tertiary amine derivative, a preparation method and an application in preparing a
plant source
fungicide, the
carvacrol tertiary amine derivative contains a cyclic secondary amine
substituent, the preparation method of the derivative is that an intermediate II is dissolved in
ethanol, then a cyclic secondary amine is added, heating and stirring are carried out,
reflux is kept, after TLC detection reaction is completed,
ethanol is removed under reduced pressure, then extraction,
water washing and purification are carried out, and the
carvacrol tertiary amine derivative is prepared. The carvacrol
tertiary amine derivative prepared by the present application exhibits obvious bacteriostatic activity on cucumber anthracnose
fungus, tomato
botrytis blight fungus, wheat scab
fungus and wheat take-all fungus. The preliminary bacteriostatic activity of carvacrol
tertiary amine derivatives 1, 3, 10 and 14 on wheat take-all fungus is 60.8%-83.2%, which is significantly better than that of
positive control hymexazol (48.6%) and reference control carvacrol (45.0%).