The invention discloses a beautifying and whitening pill and a preparation method of the beautifying and whitening pill. The pill comprises the raw materials as follows: honey, herba epimedii, Agastache rugosus, flowers carthami, almond, glossy privet fruit, radix rehmanniae preparata, Astragalus mongholicus, fructus amomi, Gorgon fruit, coix lachryma-jobi kernel and Chinese yam. The preparation method comprises the steps of (1) smashing almond, Gorgon fruit, coix lachryma-jobi kernel, Chinese yam and fructus amomi into 100-140 meshes to obtain powder A; (2) adding water into herba epimedii, Agastache rugosus, flowers carthami, glossy privet fruit, radix rehmanniae preparata and Astragalus mongholicus to decoct twice, adding 3-8 times of water by weight every time, combining a medicine liquid and concentrating to 0.4-0.6 time in weight to obtain a concentrated liquor B; and (3) mixing honey and powder A and concentrated liquor B to prepare the pill, drying till the water content is smaller than or equal to 5% by hot wind at 100-140 DEG C, sterilizing and packaging to obtain the pill. The beautifying and whitening pill is free from any chemical additives, has the functions of conditioning qi of middle-jiao energy, developing heart-yang, promoting blood circulation to remove blood stasis, removing cold and resolving dampness, and eliminating facial macula, pouch, and black eye, and beatifies and whitens rapidly.