The invention discloses a compound and application thereof in synthesis of oxidized
resveratrol derivatives in the technical field of
organic chemistry, according to a method, (E)-2-(2, 4-bis (benzyloxy) styryl)-4, 4, 5, 5-tetramethyl-1, 3, 2-dioxaborane and a halogenated
benzene compound are sequentially subjected to a
coupling reaction and a debenzylation protection reaction, and purification is performed to obtain the oxidized
resveratrol derivatives. According to the present invention, by selecting different halogenated
benzene compounds, a variety of oxidized
resveratrol derivatives with different structures are synthesized, the individual development of the synthesis
route of each product is avoided, the synthesis
route of (E)-2-(2, 4-bis (benzyloxy) styryl)-4, 4, 5, 5-tetramethyl-1, 3, 2-dioxaborane is simple, the product is easily available, the structure is simple, the industrial potential is provided, and in addition, the method can be used in the field of industrial production. Through innovative reaction steps and condition optimization, further improvement of reaction selectivity and efficiency is realized in synthesis of the oxidized resveratrol derivative, meanwhile, product stability is guaranteed, the oxidized resveratrol derivative is promoted to be converted into a mainstream functional
raw material, and large-scale production requirements can be met.